SCHEMBL5840104

SCHEMBL5840104

CCn1cnc2c(CS)nc(NCCO)nc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 16/20 0.57
TMIGD3 P0DMS9 1/20 0.50
ADORA2A P29274 1/20 0.50
ADORA2B P29275 1/20 0.50
ADORA1 P30542 1/20 0.50
CCNK O75909 2/20 0.46
CDK12 Q9NYV4 2/20 0.46
CDK2 P24941 4/20 0.43
CCNB1 P14635 3/20 0.43
CCNE1 P24864 3/20 0.43
KDM4E B2RXH2 1/20 0.41
CCNB2 O95067 1/20 0.41
CCNE2 O96020 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
GAA P10253 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5839632 0.83 CDK1 (0.71) CDK1CCNKCDK12CDK2CCNB1
SCHEMBL27397625 0.82 CDK1 (0.57) CDK1TMIGD3ADORA2AADORA2BADORA1
SCHEMBL5840099 0.79 CDK1 (0.56) CDK1TMIGD3ADORA2AADORA2BADORA1
SCHEMBL5840230 0.74 CDK1 (0.82) CDK1CCNKCDK12PRKCA
SCHEMBL5840633 0.74 CDK1 (0.50) CDK1TMIGD3ADORA2AADORA2BADORA1
SCHEMBL5839924 0.73 CDK1 (1.00) CDK1CDK5CDK5R1PRKCA
SCHEMBL18520823 0.73 CDK1 (0.53) CDK1TMIGD3ADORA2AADORA2BADORA1
SCHEMBL12982866 0.72 CDK1 (0.81) CDK1CDK2CCNE1CCNE2ALDH1A1
SCHEMBL5839245 0.72 CDK1 (0.81) CDK1CCNKCDK12CDK5CDK5R1
SCHEMBL5840277 0.72 CDK1 (0.71) CDK1CCNKCDK12CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7091346-B1 Purine derivatives and processes for their preparation NOVARTIS AG (CH) 2006-08-15 US disclosed
EP-0874846-B1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 2003-04-02 EP disclosed
EP-0874846-A1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION Novartis AG (CH) 1998-11-04 EP disclosed
WO-1997016452-A1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 1997-05-09 WO disclosed