SCHEMBL5840422

SCHEMBL5840422

CC(=O)Nc1ncc(-c2ccccc2)s1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.72
GSTO1 P78417 1/20 0.67
CCNE1 P24864 3/20 0.65
CDK2 P24941 3/20 0.65
CDK5 Q00535 2/20 0.65
SCD O00767 1/20 0.65
ACP1 P24666 1/20 0.62
CNR1 P21554 1/20 0.60
MKNK1 Q9BUB5 1/20 0.60
FFAR2 O15552 1/20 0.56
CYP1A2 P05177 1/20 0.55
MAPK1 P28482 1/20 0.55
APOBEC3A P31941 1/20 0.55
APOBEC3G Q9HC16 1/20 0.55
LIMK1 P53667 1/20 0.54
CCNE2 O96020 1/20 0.53
WNT3A P56704 1/20 0.52
NQO2 P16083 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30142626 0.85 KDR (0.65) KDRGSTO1CCNE1CDK2CDK5
SCHEMBL24074022 0.85 KDR (0.65) KDRGSTO1CCNE1CDK2CDK5
SCHEMBL17632040 0.84 ABL1 (0.62) KDRGSTO1CCNE1CDK2CDK5
SCHEMBL17014785 0.84 KDR (0.68) KDRGSTO1CCNE1CDK2CDK5
SCHEMBL10252594 0.84 KDR (1.00) KDRGSTO1CCNE1CDK2CDK5
SCHEMBL2256136 0.84 KDR (0.72) KDRGSTO1CCNE1CDK2CDK5
SCHEMBL12496031 0.82 KDR (0.50) KDRGSTO1CCNE1CDK2CDK5
SCHEMBL7518296 0.81 KDR (0.50) KDRGSTO1CCNE1CDK2CDK5
SCHEMBL6281775 0.81 CNR1 (0.82) KDRGSTO1CCNE1CDK2CDK5
SCHEMBL69753 0.81 CCNE1 (0.74) KDRGSTO1CCNE1CDK2CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102725287-B 1,3, 4-oxadiazole-2-carboxamide compounds PHARMA IP GENERAL INC ASS 2015-07-01 CN disclosed
CN-102725287-A 1,3, 4-oxadiazole-2-carboxamide compounds PHARMA IP GENERAL INC ASS 2012-10-10 CN disclosed
US-7037929-B1 2-amino-thiazole derivatives, process for their preparation, and their use as antitumor agents PHARMACIA & UPJOHN S.P.A. (IT) 2006-05-02 US disclosed
EP-1124810-B9 2-AMINO-THIAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND THEIR USE AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-12-28 EP disclosed
EP-1124810-B1 2-AMINO-THIAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND THEIR USE AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-05-04 EP disclosed