SCHEMBL5840470

SCHEMBL5840470

[c]1ncc(-c2ccnc(-c3ccccc3)n2)c(-c2ccccc2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
KMT2A Q03164 5/20 0.39
MEN1 O00255 4/20 0.39
MAPT P10636 3/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
KDM4E B2RXH2 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
POLB P06746 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
PTK2B Q14289 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ADORA2A P29274 3/20 0.36
AURKA O14965 1/20 0.36
HSP90AA1 P07900 1/20 0.36
PRKACA P17612 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4316992 0.83 CYP2A6 (0.36) MAPTNPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL3575254 0.77 ADORA1 (0.39) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL16060090 0.72 KDM4E (0.42) MAPTNPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL29620532 0.71 AURKA (0.63) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL190954 0.71 AURKA (0.63) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL558261 0.71 AKT1 (0.35)
SCHEMBL31074804 0.70 GABRA1 (0.49) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7358193 0.70 CYP2A6 (0.57) NPC1RAB9AKDM4ESMN1; SMN2POLB
Ammonia Solution, Strong SCHEMBL20267253 0.69 AURKA (0.61) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL18952722 0.69 KDM4E (0.47) KMT2AMEN1NPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7019026-B1 Modulators of Protein Tyrosine Phosphatases (PTPases) NOVO NORDISK A/S (DK) 2006-03-28 US disclosed