SCHEMBL5840596

SCHEMBL5840596

CCn1cnc2c(Nc3ccc(Cl)c(C(F)(F)F)c3)nc(NCCO)nc21

nearest known ligand 0.70

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 17/20 0.70
PRKCA P17252 5/20 0.58
CDK5 Q00535 2/20 0.57
CDK5R1 Q15078 2/20 0.57
CCNB1 P14635 1/20 0.52
EIF2AK2 P19525 1/20 0.52
GSK3B P49841 1/20 0.52
MERTK Q12866 1/20 0.52
NPC1 O15118 1/20 0.50
CCNK O75909 1/20 0.49
CDK12 Q9NYV4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5839982 0.91 CDK1 (0.71) CDK1PRKCACDK5CDK5R1CCNB1
SCHEMBL5839952 0.85 CDK5 (0.56) CDK1PRKCACDK5CDK5R1CCNB1
SCHEMBL5839936 0.85 CDK5 (0.56) CDK1PRKCACDK5CDK5R1CCNB1
SCHEMBL5839245 0.84 CDK1 (0.81) CDK1PRKCACDK5CDK5R1CCNK
SCHEMBL5840868 0.84 YTHDC1 (0.52) CDK1PRKCANPC1
SCHEMBL5839355 0.83 CDK1 (1.00) CDK1PRKCACDK5CDK5R1CCNB1
SCHEMBL5840277 0.82 CDK1 (0.71) CDK1PRKCACDK5CDK5R1NPC1
SCHEMBL5839924 0.82 CDK1 (1.00) CDK1PRKCACDK5CDK5R1NPC1
SCHEMBL5840457 0.81 CDK1 (0.73) CDK1PRKCACCNB1
SCHEMBL5840462 0.81 CDK1 (0.73) CDK1PRKCACCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7091346-B1 Purine derivatives and processes for their preparation NOVARTIS AG (CH) 2006-08-15 US disclosed
EP-0874846-B1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 2003-04-02 EP disclosed
CN-1066147-C Purine derivatives and process for preparing same 诺瓦提斯公司 2001-05-23 CN disclosed
CN-1202896-A Purine derivatives and processes for their preparation 诺瓦提斯公司 1998-12-23 CN disclosed
EP-0874846-A1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION Novartis AG (CH) 1998-11-04 EP disclosed
WO-1997016452-A1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 1997-05-09 WO disclosed