SCHEMBL58410

SCHEMBL58410

N[C@@H](CS)C(=O)Oc1cccs1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 2/20 0.40
MMP1 P03956 1/20 0.40
MMP9 P14780 1/20 0.40
MMP12 P39900 1/20 0.40
SLC1A3 P43003 1/20 0.37
SLC1A2 P43004 1/20 0.37
SLC1A1 P43005 1/20 0.37
KMT2A Q03164 2/20 0.36
MAPT P10636 1/20 0.36
ADAM17 P78536 1/20 0.36
ATM Q13315 1/20 0.36
KIF11 P52732 1/20 0.36
POLB P06746 3/20 0.36
ALDH1A1 P00352 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PTGS1 P23219 1/20 0.34
SLC7A11 Q9UPY5 1/20 0.34
ADRA2A P08913 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8430877 0.88 MMP1 (0.38) MMP2MMP1MMP9MMP12SLC1A3
SCHEMBL2009145 0.85 MMP1 (0.41) MMP2MMP1MMP9MMP12SLC1A3
SCHEMBL4350616 0.83 KIF11 (0.41) MMP2MMP1MMP9MMP12SLC1A3
SCHEMBL28535887 0.82 KIF11 (0.36) MMP2MMP1MMP9MMP12SLC1A3
SCHEMBL1897993 0.81 MMP1 (0.41) MMP2MMP1MMP9MMP12SLC1A3
SCHEMBL9878919 0.81 KIF11 (0.40) MMP2MMP1MMP9MMP12SLC1A3
SCHEMBL5680233 0.80 ALPI (0.51) SLC1A3SLC1A2SLC1A1PTGS1CTSC
SCHEMBL29159324 0.80 MMP1 (0.40) MMP2MMP1MMP9MMP12SLC1A3
SCHEMBL5801530 0.79 DPP7 (0.42) MMP2MMP1MMP9MMP12SLC1A3
SCHEMBL3399442 0.78 MMP1 (0.43) MMP2MMP1MMP9MMP12SLC1A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 8567 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260146088-A1 ANTI-CD79B ANTIBODIES AND IMMUNOCONJUGATES AND METHODS OF USE GENENTECH, INC. (US) 2026-05-28 US claimed
US-20260137794-A1 LIGAND-DRUG CONJUGATE AND USE THEREOF SYSTIMMUNE INC (US) 2026-05-21 US claimed
US-20260137630-A1 COMPOSITIONS AND METHODS FOR T CELL TARGETED DELIVERY OF THERAPEUTIC AGENTS AND ACTIVATION OF T CELLS THE TRUSTEES OF THE UNIV OF PENNSYLVANIA (US) 2026-05-21 US claimed
CN-122011005-A Use of tris (trimethylsilyl) silane in disulfide hydrosilation reactions 中山大学 2026-05-12 CN claimed
WO-2026090156-A1 1,3,5-TRIAZINANE-2,4,6-TRIONE-DERIVED IONIZABLE LIPID COMPOUNDS AND LIPID NANOPARTICLES (LNPS) COMPRISING THE SAME THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2026-04-30 WO claimed
EP-4637833-A2 CEREBLON DEGRADER CONJUGATES, AND USES THEREOF Genentech, Inc. (US) 2025-10-29 EP claimed
US-12440706-B2 Conjugated chemical inducers of degradation and methods of use GENENTECH, INC. (US) 2025-10-14 US claimed
WO-2025134068-A1 ANTIBODY DRUG CONJUGATES TARGETING PROTEINOPATHIES, AND USES THEREOF AC IMMUNE SA (CH) 2025-06-26 WO claimed
US-12296018-B2 Albumin binding peptide-drug (AlBiPeD) conjugates and methods of making and using same DUKE UNIVERSITY (US) 2025-05-13 US claimed
US-20250145575-A1 MACROMOLECULE-SUPPORTED 8-SULFONYL-BENZAZEPINE COMPOUNDS AND THEIR USES BOLT BIOTHERAPEUTICS, INC. (US) 2025-05-08 US claimed
EP-0474789-B1 CYSTEINE THIOL-PROTECTED PEPTIDES FOR USE IN IMMUNOASSAYS GENETIC SYSTEMS CORP (US) 1998-01-28 EP claimed
WO-1997031944-A1 FRAGMENTS OF CR1 AND THEIR USE ADPROTECH PLC (GB) 1997-09-04 WO claimed
WO-1997004004-A1 CYSTEINE PROTEASE INHIBITORS FOR USE IN TREATMENT OF IgE MEDIATED ALLERGIC DISEASES PEPTIDE THERAPEUTICS LIMITED (GB) 1997-02-06 WO claimed
US-5439792-A Synthesizing a cyclic viral protein epitope GENETIC SYSTEMS CORPORATION (US) 1995-08-08 US claimed
EP-0474789-A4 CYSTEINE THIOL-PROTECTED PEPTIDES FOR USE IN IMMUNOASSAYS 1992-06-03 EP claimed
EP-0474789-A1 CYSTEINE THIOL-PROTECTED PEPTIDES FOR USE IN IMMUNOASSAYS GENETIC SYSTEMS CORPORATION (US) 1992-03-18 EP claimed
EP-0233973-B1 MIXTURE OF AMINO ACID DERIVATIVES, PROCESS OF PRODUCING THE MIXTURE AND USE OF THE MIXTURE FOR QUANTITATIVE DETERMINATION OF THE AMINO ACIDS Hewlett-Packard GmbH (DE) 1990-12-27 EP claimed
WO-1990015071-A1 CYSTEINE THIOL-PROTECTED PEPTIDES FOR USE IN IMMUNOASSAYS GENETIC SYSTEMS CORPORATION (US) 1990-12-13 WO claimed
EP-0233973-A1 Mixture of amino acid derivatives, process of producing the mixture and use of the mixture for quantitative determination of the amino acids Hewlett-Packard GmbH (DE) 1987-09-02 EP claimed
EP-0105525-B1 THIOHYDRAZINE-1,2-DICARBONIC ACIDS, PROCESS FOR THEIR PREPARATION AND THEIR USE Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 1986-09-10 EP claimed