SCHEMBL5847112

SCHEMBL5847112

Cc1ccc(C)n1CCCCN1CC=C(c2ccccc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.59
HTR1A P08908 1/20 0.52
PARP1 P09874 2/20 0.52
HTR7 P34969 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5848153 0.99 SIGMAR1 (0.57) SIGMAR1HTR1APARP1HTR7
SCHEMBL5846215 0.86 SIGMAR1 (0.63) SIGMAR1HTR1APARP1HTR7
Hydrochloric Acid SCHEMBL5847569 0.85 SIGMAR1 (0.62) SIGMAR1HTR1APARP1HTR7
SCHEMBL256663 0.84 SIGMAR1 (0.63) SIGMAR1HTR1APARP1
SCHEMBL14601668 0.82 SIGMAR1 (0.60) SIGMAR1HTR1A
SCHEMBL7297566 0.81 SIGMAR1 (0.63) SIGMAR1HTR1APARP1
SCHEMBL5544346 0.81 SIGMAR1 (0.63) SIGMAR1HTR1APARP1
SCHEMBL6160767 0.80 SIGMAR1 (0.53) SIGMAR1PARP1
Hydrochloric Acid SCHEMBL7299927 0.79 SIGMAR1 (0.61) SIGMAR1HTR1APARP1
SCHEMBL5846286 0.79 SIGMAR1 (0.61) SIGMAR1HTR1APARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39113-E1 Utilization of derivatives of tetrahydropyridines(or 4-hydroxypiperidines)-butylazols in the preparation of a medicament for the treatment of pain LABORATORIES DEL DR. ESTEVE, S.A. (ES) 2006-05-30 US claimed
EP-1097698-B1 UTILIZATION OF DERIVATIVES OF TETRAHYDROPYRIDINES (OR 4-HYDROXYPIPERIDINES)-BUTYLAZOLS IN THE PREPARATION OF A MEDICAMENT FOR THE TREATMENT OF PAIN ESTEVE LABOR DR (ES) 2003-05-07 EP claimed
US-6384055-B1 ANALGESICS LABORATORIOS DEL DR. ESTEVES, S.A. (ES) 2002-05-07 US claimed
EP-1097698-A2 UTILIZATION OF DERIVATIVES OF TETRAHYDROPYRIDINES (OR 4-HYDROXYPIPERIDINES)-BUTYLAZOLS IN THE PREPARATION OF A MEDICAMENT FOR THE TREATMENT OF PAIN LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2001-05-09 EP claimed