SCHEMBL5847206

SCHEMBL5847206

CC(C)(C)OC(=O)N1CC[C@H]2[C@@H](C1)c1cc(-c3ccc(C(F)(F)F)cc3Cl)cc3c1N2CCCC3

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.42
HTR2C P28335 3/20 0.42
HTR2B P41595 1/20 0.42
GPR119 Q8TDV5 4/20 0.40
ALK Q9UM73 2/20 0.37
TACR1 P25103 1/20 0.36
MC4R P32245 1/20 0.36
P2RY14 Q15391 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
PDK2 Q15119 2/20 0.35
MCL1 Q07820 1/20 0.35
MAPT P10636 1/20 0.35
STS P08842 1/20 0.35
RORC P51449 1/20 0.34
DRD2 P14416 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5848017 0.98 HTR2A (0.45) HTR2AHTR2CHTR2BGPR119ALK
SCHEMBL5847844 0.94 GPR119 (0.42) HTR2AHTR2CHTR2BGPR119ALK
SCHEMBL5849172 0.91 HTR2A (0.50) HTR2AHTR2CHTR2BGPR119ALK
SCHEMBL5847375 0.90 CNR1 (0.40) HTR2AHTR2CHTR2BGPR119NPC1
SCHEMBL5847589 0.89 HTR2A (0.53) HTR2AHTR2CHTR2BGPR119ALK
SCHEMBL5428406 0.89 HTR2C (0.42) HTR2AHTR2CHTR2BPDK2MAPT
SCHEMBL5847743 0.88 HTR2A (0.48) HTR2AHTR2CHTR2BGPR119NPC1
SCHEMBL5847225 0.88 MEN1 (0.39) HTR2AHTR2CHTR2BGPR119NPC1
SCHEMBL5848567 0.88 HTR2C (0.41) HTR2AHTR2CHTR2BGPR119NPC1
SCHEMBL5635408 0.86 GPR119 (0.39) GPR119ALKTACR1MC4RP2RY14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed