SCHEMBL5847735

SCHEMBL5847735

COC(CN)c1ccccc1Br

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.42
ALDH1A1 P00352 2/20 0.42
CYP3A4 P08684 1/20 0.42
ALOX15 P16050 1/20 0.42
IDO1 P14902 3/20 0.41
TDO2 P48775 1/20 0.41
CYP2C9 P11712 1/20 0.40
AOC3 Q16853 1/20 0.38
HTT P42858 1/20 0.36
TAAR1 Q96RJ0 3/20 0.35
NISCH Q9Y2I1 1/20 0.33
HTR2A P28223 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
OPRL1 P41146 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10860608 0.77 IDO1 (0.47) ALDH1A1CYP3A4IDO1TDO2CYP2C9
SCHEMBL5847586 0.74 TAAR1 (0.50) CYP2C19ALDH1A1CYP3A4ALOX15IDO1
Iodide SCHEMBL25290234 0.73 AOC3 (0.65) CYP2C19ALDH1A1CYP2C9AOC3HTR2A
SCHEMBL20970894 0.73 HTR2A (0.49) TAAR1HTR2A
SCHEMBL29543232 0.73 HTR2A (0.49) TAAR1HTR2A
SCHEMBL1471049 0.73 IDO1 (0.42) ALDH1A1IDO1TDO2HTTTAAR1
SCHEMBL6325 0.73 CYP2C19 (0.44) CYP2C19ALDH1A1CYP3A4ALOX15IDO1
SCHEMBL11111739 0.73 IDO1 (0.42) ALDH1A1IDO1TDO2HTTTAAR1
SCHEMBL29369499 0.73 CYP2C19 (0.44) CYP2C19ALDH1A1CYP3A4ALOX15IDO1
SCHEMBL20773755 0.72 ALOX12 (0.37) IDO1TDO2AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7078567-B2 Amination process JOHNSTON JEFFREY N 2006-07-18 US disclosed
US-20040082778-A1 Amination process JOHNSTON JEFFREY N (US) 2004-04-29 US disclosed
US-6670479-B2 An sp2 hybridized radical is reacted with an azomethine group to form pyrrolidine and indole compounds ADVANCED RESEARCH AND TECHNOLOGY INSTITUTE, INC. 2003-12-30 US disclosed
WO-2002072547-A1 AMINATION PROCESS ADVANCED RESEARCH AND TECHNOLOGY INSTITUTE, INC. (US) 2002-09-19 WO disclosed
US-20020128490-A1 Amination process ADVANCED RESEARCH AND TECHNOLOGY INSTITUTE, INC. 2002-09-12 US disclosed
WO-2002070439-A2 AMINATION PROCESS JOHNSTON, JEFFREY, N. 2002-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040082778-A1 Amination process IDO2, INMT, IDO1 CYP2C19 1254/4885ALDH1A1 567/4885CYP3A4 122/4885
US-20020128490-A1 Amination process IDO2, INMT, IDO1 CYP2C19 1146/4885ALDH1A1 106/4885CYP3A4 93/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.