SCHEMBL5847802

SCHEMBL5847802

CC(C)Oc1ccc(-c2cc3c4c(c2)[C@@H]2CN(C(=O)OC(C)(C)C)CC[C@@H]2N4CCCC3)c(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.53
HTR2C P28335 4/20 0.53
HTR2B P41595 1/20 0.53
GPR119 Q8TDV5 4/20 0.38
EPHX2 P34913 1/20 0.37
S1PR1 P21453 1/20 0.35
S1PR3 Q99500 1/20 0.35
USP30 Q70CQ3 1/20 0.34
LIPE Q05469 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
DRD2 P14416 2/20 0.33
SFRP1 Q8N474 2/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
TACR1 P25103 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5848817 0.98 HTR2A (0.56) HTR2AHTR2CHTR2BGPR119EPHX2
SCHEMBL5847472 0.95 HTR2A (0.49) HTR2AHTR2CHTR2BGPR119EPHX2
SCHEMBL5847212 0.92 HTR2A (0.63) HTR2AHTR2CHTR2BGPR119EPHX2
SCHEMBL5421842 0.91 HTR2A (0.56) HTR2AHTR2CHTR2BS1PR1S1PR3
SCHEMBL5416044 0.90 HTR2A (0.66) HTR2AHTR2CHTR2BGPR119EPHX2
SCHEMBL5848217 0.90 HTR2A (0.66) HTR2AHTR2CHTR2BGPR119EPHX2
SCHEMBL5849172 0.89 HTR2A (0.50) HTR2AHTR2CHTR2BGPR119EPHX2
SCHEMBL5848926 0.89 HTR2A (0.50) HTR2AHTR2CHTR2BGPR119NPC1
SCHEMBL5410701 0.88 HTR2A (0.59) HTR2AHTR2CHTR2BS1PR1S1PR3
SCHEMBL5848068 0.88 HTR2A (0.65) HTR2AHTR2CHTR2BGPR119EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed