SCHEMBL5848926

SCHEMBL5848926

CC(C)(C)OC(=O)N1CC[C@H]2[C@@H](C1)c1cc(-c3ccc(F)cc3C(F)(F)F)cc3c1N2CCCC3

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 8/20 0.50
HTR2C P28335 8/20 0.50
HTR2B P41595 1/20 0.50
DRD2 P14416 4/20 0.40
GPR119 Q8TDV5 2/20 0.39
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
BRD3 Q15059 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HTR1A P08908 1/20 0.36
DRD4 P21917 1/20 0.36
SLC6A4 P31645 1/20 0.36
PAK1 Q13153 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5849629 0.98 HTR2A (0.53) HTR2AHTR2CHTR2BDRD2GPR119
SCHEMBL5849172 0.92 HTR2A (0.50) HTR2AHTR2CHTR2BDRD2GPR119
SCHEMBL5847212 0.91 HTR2A (0.63) HTR2AHTR2CHTR2BGPR119
SCHEMBL5846925 0.90 HTR2A (0.47) HTR2AHTR2CHTR2BDRD2GPR119
SCHEMBL5847589 0.90 HTR2A (0.53) HTR2AHTR2CHTR2BGPR119NPC1
SCHEMBL5847802 0.89 HTR2A (0.53) HTR2AHTR2CHTR2BDRD2GPR119
SCHEMBL5846988 0.89 HTR2A (0.47) HTR2AHTR2CHTR2BGPR119HDAC1
SCHEMBL5413963 0.88 HTR2A (0.50) HTR2AHTR2CHTR2BDRD2HTR1A
SCHEMBL5848217 0.88 HTR2A (0.66) HTR2AHTR2CHTR2BGPR119
SCHEMBL5416044 0.88 HTR2A (0.66) HTR2AHTR2CHTR2BGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed