SCHEMBL5847872

SCHEMBL5847872

COc1ccc(C(C)C)cc1-c1cc2c3c(c1)[C@H]1CN(C(=O)OC(C)(C)C)CC[C@H]1N3CC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 9/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
PIK3CD O00329 2/20 0.37
PIK3CA P42336 2/20 0.37
PIK3CB P42338 2/20 0.37
PIK3CG P48736 2/20 0.37
GPR119 Q8TDV5 1/20 0.37
CCR3 P51677 1/20 0.37
USP30 Q70CQ3 1/20 0.36
STS P08842 1/20 0.36
CCNT1 O60563 2/20 0.35
CDK9 P50750 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5848229 0.94 NPC1 (0.40) PDE4BNPC1ALDH1A1MAPTMAPK1
SCHEMBL5418618 0.89 CCR3 (0.39) PDE4BCCR3HTR2AHTR2CHTR2B
SCHEMBL5418614 0.89 CCR3 (0.39) PDE4BCCR3HTR2AHTR2CHTR2B
SCHEMBL5635435 0.85 PDE4B (0.39) PDE4BNPC1ALDH1A1MAPTMAPK1
SCHEMBL5847917 0.85 HTR2A (0.46) PDE4BALDH1A1MAPTHTTMEN1
SCHEMBL5847910 0.85 PIK3CD (0.49) PDE4BPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL5846970 0.84 HTR2A (0.43) ALDH1A1HTTMEN1KMT2AGPR119
SCHEMBL5420299 0.83 CCR3 (0.39) ALDH1A1CCR3HTR2AHTR2CHTR2B
SCHEMBL5420302 0.83 CCR3 (0.39) ALDH1A1CCR3HTR2AHTR2CHTR2B
SCHEMBL5849353 0.81 GPR119 (0.37) PDE4BPIK3CDPIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US claimed
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed