SCHEMBL5850607

SCHEMBL5850607

Cc1ccc(S(=O)(=O)N(C)C2(C(=O)N[C@@H](Cc3ccc(OC4CCN(C)CC4)cc3)C(=O)O)CCCC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 16/20 0.47
ITGB1 P05556 15/20 0.47
ITGB7 P26010 9/20 0.45
ALDH1A1 P00352 1/20 0.42
TDP1 Q9NUW8 1/20 0.40
ACACB O00763 1/20 0.39
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5852314 0.94 ITGB1 (0.40) ITGA4ITGB1ITGB7ALDH1A1ACACB
SCHEMBL5850996 0.92 ITGA4 (0.39) ITGA4ITGB1ITGB7ALDH1A1ACACB
SCHEMBL5850857 0.83 ITGB1 (0.64) ITGA4ITGB1ITGB7ALDH1A1TDP1
SCHEMBL5850545 0.82 ITGB1 (0.52) ITGA4ITGB1ITGB7TDP1
SCHEMBL7401948 0.81 ITGB1 (0.61) ITGA4ITGB1ITGB7ALDH1A1TDP1
SCHEMBL7328129 0.78 ITGA4 (0.63) ITGA4ITGB1ITGB7ALDH1A1
SCHEMBL5851039 0.78 ATM (0.55) ITGA4ITGB1ITGB7ALDH1A1
SCHEMBL5850976 0.76 ITGB1 (0.47) ITGA4ITGB1ITGB7ALDH1A1TDP1
SCHEMBL7409938 0.76 ATM (0.55) ITGA4ITGB1ITGB7ALDH1A1
SCHEMBL5850641 0.76 ITGB1 (0.44) ITGA4ITGB1ITGB7ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7030114-B1 Compounds which inhibit leukocyte adhesion mediated by VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2006-04-18 US disclosed
EP-0994895-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-04-26 EP disclosed
WO-1999006435-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO disclosed