SCHEMBL5850976

SCHEMBL5850976

Cc1ccc(S(=O)(=O)N(C)C2(C(=O)N[C@@H](Cc3ccc(NC(=O)C4CCNCC4)cc3)C(=O)O)CCCC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 12/20 0.47
ITGA4 P13612 12/20 0.47
ALDH1A1 P00352 1/20 0.44
ITGB7 P26010 2/20 0.43
TDP1 Q9NUW8 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MMP9 P14780 1/20 0.40
USP30 Q70CQ3 1/20 0.40
ENPP3 O14638 1/20 0.39
ENPP1 P22413 1/20 0.39
ENPP2 Q13822 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5850857 0.83 ITGB1 (0.64) ITGB1ITGA4ALDH1A1ITGB7TDP1
SCHEMBL7401948 0.81 ITGB1 (0.61) ITGB1ITGA4ALDH1A1ITGB7TDP1
SCHEMBL5850609 0.81 MMP9 (0.49) ITGB1ITGA4ALDH1A1ITGB7TDP1
SCHEMBL5852274 0.79 ITGB1 (0.51) ITGB1ITGA4ITGB7MMP9
SCHEMBL5850463 0.79 PTPN2 (0.46) ALDH1A1LMNA
SCHEMBL5850545 0.77 ITGB1 (0.52) ITGB1ITGA4ITGB7TDP1
SCHEMBL5691025 0.77 ITGB1 (0.63) ITGB1ITGA4ALDH1A1ITGB7
SCHEMBL5850607 0.76 ITGA4 (0.47) ITGB1ITGA4ALDH1A1ITGB7TDP1
SCHEMBL5850632 0.76 ALDH1A1 (0.41) ITGB1ITGA4ALDH1A1LMNAHTT
SCHEMBL5851039 0.76 ATM (0.55) ITGB1ITGA4ALDH1A1ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7030114-B1 Compounds which inhibit leukocyte adhesion mediated by VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2006-04-18 US disclosed
EP-0994895-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-04-26 EP disclosed
WO-1999006435-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO disclosed