SCHEMBL5850823

SCHEMBL5850823

CCOC(=O)[C@H](Cc1ccc(OC(=O)N(C)C)cc1)NC(=O)C1(N(C)S(=O)(=O)c2ccc(C)cc2)CCCC1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 9/20 0.42
ITGA4 P13612 9/20 0.42
ITGB7 P26010 1/20 0.39
PTGES O14684 1/20 0.37
ATM Q13315 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
KMT2A Q03164 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
BACE1 P56817 1/20 0.35
NPSR1 Q6W5P4 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5850641 0.95 ITGB1 (0.44) ITGB1ITGA4ITGB7PTGESATM
SCHEMBL5850545 0.91 ITGB1 (0.52) ITGB1ITGA4ITGB7PTGESTDP1
SCHEMBL5850329 0.91 ITGB1 (0.41) ITGB1ITGA4ITGB7PTGESATM
SCHEMBL5850996 0.83 ITGA4 (0.39) ITGB1ITGA4ITGB7L3MBTL1NPSR1
SCHEMBL5851039 0.83 ATM (0.55) ITGB1ITGA4ITGB7ATML3MBTL1
SCHEMBL7409938 0.81 ATM (0.55) ITGB1ITGA4ITGB7ATML3MBTL1
SCHEMBL5850926 0.80 ALDH1A1 (0.45) ITGB1ITGA4KMT2ANPSR1LMNA
SCHEMBL5850857 0.79 ITGB1 (0.64) ITGB1ITGA4ITGB7TDP1
SCHEMBL5852314 0.78 ITGB1 (0.40) ITGB1ITGA4ITGB7ATML3MBTL1
SCHEMBL7401948 0.77 ITGB1 (0.61) ITGB1ITGA4ITGB7TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994895-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-04-26 EP claimed
WO-1999006435-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO claimed
US-7030114-B1 Compounds which inhibit leukocyte adhesion mediated by VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2006-04-18 US disclosed
EP-0994895-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-04-26 EP disclosed
WO-1999006435-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO disclosed