SCHEMBL5852256

SCHEMBL5852256

Fc1ccc(-c2nn(C(c3ccccc3)(c3ccccc3)C3C=CC=CC3)cc2-c2ccc3ncn(-c4ccc(F)cc4)c3c2)cc1

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ATM Q13315 6/20 0.32
SRC P12931 1/20 0.32
BRAF P15056 1/20 0.32
KDR P35968 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
MAPK10 P53779 1/20 0.31
NCOA1 Q15788 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31
FGFR1 P11362 1/20 0.31
CDK9 P50750 1/20 0.30
PIK3R2 O00459 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3846716 0.91 POLB (0.33) PIK3R2
SCHEMBL3847150 0.86 FGFR1 (0.33) FGFR1
SCHEMBL3846777 0.85 ATM (0.36) ATMKDRALDH1A1HPGDMAPK1
SCHEMBL3847835 0.84 ALOX5AP (0.37) ALDH1A1HPGD
SCHEMBL3847729 0.83 PIK3CD (0.34) ALDH1A1HPGDMAPK1
SCHEMBL3855066 0.82 ALDH1A1 (0.32) ALDH1A1MAPK1
SCHEMBL3847279 0.82 CCR3 (0.36) ALDH1A1HPGD
SCHEMBL3845877 0.82
SCHEMBL5852255 0.82 SRC (0.38) ATMSRCBRAFKDRALDH1A1
SCHEMBL3856288 0.81 CNR1 (0.34) CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7074801-B1 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof EISAI CO., LTD. (JP) 2006-07-11 US disclosed
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed