SCHEMBL5852432

SCHEMBL5852432

C=CCOCCc1ccc(OC[C@@H](O)CNC(C)C)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.73
ADRB1 P08588 4/20 0.70
ADRB2 P07550 3/20 0.70
NR3C1 P04150 1/20 0.70
ADRA1A P35348 1/20 0.70
CYP2J2 P51589 1/20 0.70
PDE4D Q08499 1/20 0.70
LMNA P02545 2/20 0.67
MEN1 O00255 1/20 0.67
CYP1A2 P05177 1/20 0.67
CYP2C9 P11712 1/20 0.67
KMT2A Q03164 1/20 0.67
GAA P10253 1/20 0.65
BLM P54132 1/20 0.65
TMEM97 Q5BJF2 1/20 0.65
SIGMAR1 Q99720 1/20 0.65
NPY1R P25929 1/20 0.60
NPY2R P49146 1/20 0.60
PMP22 Q01453 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5351511 1.00 CYP2D6 (0.73) CYP2D6ADRB1ADRB2NR3C1ADRA1A
SCHEMBL7307918 0.88 CYP2D6 (0.76) CYP2D6ADRB1ADRB2NR3C1ADRA1A
SCHEMBL10739631 0.85 ADRB1 (0.76) CYP2D6ADRB1ADRB2NR3C1ADRA1A
SCHEMBL11856247 0.85 ADRB1 (0.76) CYP2D6ADRB1ADRB2NR3C1ADRA1A
SCHEMBL220354 0.85 ADRB1 (0.76) CYP2D6ADRB1ADRB2NR3C1ADRA1A
SCHEMBL11854073 0.85 CYP2D6 (1.00) CYP2D6ADRB1ADRB2ADRA1ALMNA
Hydrochloric Acid SCHEMBL11853087 0.83 CYP2D6 (0.97) CYP2D6ADRB1ADRB2ADRA1ALMNA
SCHEMBL28407475 0.83 ADRB1 (0.73) CYP2D6ADRB1ADRB2NR3C1ADRA1A
Metoprolol SCHEMBL1561123 0.82 ADRB1 (1.00) CYP2D6ADRB1ADRB2NR3C1ADRA1A
Metoprolol SCHEMBL4093 0.82 ADRB1 (1.00) CYP2D6ADRB1ADRB2NR3C1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6989465-B1 S-(−)-1-{4-[2-(allyloxy)-ethyl]phenoxy}-3-isopropylamino propan-2-ol, process for preparation thereof and process for preparation of S-(−)betaxolo COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2006-01-24 US claimed
US-6989465-B1 S-(−)-1-{4-[2-(allyloxy)-ethyl]phenoxy}-3-isopropylamino propan-2-ol, process for preparation thereof and process for preparation of S-(−)betaxolo COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2006-01-24 US disclosed
US-6989465-B1 S-(−)-1-{4-[2-(allyloxy)-ethyl]phenoxy}-3-isopropylamino propan-2-ol, process for preparation thereof and process for preparation of S-(−)betaxolo COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2006-01-24 US disclosed
US-6989465-B1 S-(−)-1-{4-[2-(allyloxy)-ethyl]phenoxy}-3-isopropylamino propan-2-ol, process for preparation thereof and process for preparation of S-(−)betaxolo COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2006-01-24 US disclosed