SCHEMBL220354

SCHEMBL220354

CC(C)NCC(O)COc1ccc(CCOCO)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 5/20 0.76
ADRB2 P07550 4/20 0.76
CYP2D6 P10635 2/20 0.76
NR3C1 P04150 1/20 0.76
ADRA1A P35348 1/20 0.76
CYP2J2 P51589 1/20 0.76
PDE4D Q08499 1/20 0.76
LMNA P02545 2/20 0.72
MEN1 O00255 1/20 0.72
CYP1A2 P05177 1/20 0.72
CYP2C9 P11712 1/20 0.72
KMT2A Q03164 1/20 0.72
GAA P10253 1/20 0.71
BLM P54132 1/20 0.71
TMEM97 Q5BJF2 1/20 0.71
SIGMAR1 Q99720 1/20 0.71
NPY1R P25929 1/20 0.65
NPY2R P49146 1/20 0.65
PMP22 Q01453 1/20 0.65
NPSR1 Q6W5P4 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11856247 0.90 ADRB1 (0.76) ADRB1ADRB2CYP2D6NR3C1ADRA1A
SCHEMBL10739631 0.90 ADRB1 (0.76) ADRB1ADRB2CYP2D6NR3C1ADRA1A
SCHEMBL28407475 0.87 ADRB1 (0.73) ADRB1ADRB2CYP2D6NR3C1ADRA1A
(S)-Metoprolol SCHEMBL121589 0.86 ADRB1 (1.00) ADRB1ADRB2CYP2D6NR3C1ADRA1A
Metoprolol SCHEMBL1561123 0.86 ADRB1 (1.00) ADRB1ADRB2CYP2D6NR3C1ADRA1A
Metoprolol SCHEMBL4093 0.86 ADRB1 (1.00) ADRB1ADRB2CYP2D6NR3C1ADRA1A
(R)-Metoprolol SCHEMBL40918 0.86 ADRB1 (1.00) ADRB1ADRB2CYP2D6NR3C1ADRA1A
SCHEMBL3462992 0.86 ADRB2 (0.75) ADRB1ADRB2CYP2D6NR3C1ADRA1A
(S)-Metoprolol SCHEMBL2638035 0.85 ADRB1 (0.97) ADRB1ADRB2CYP2D6NR3C1ADRA1A
(S)-Metoprolol SCHEMBL6728301 0.85 ADRB1 (0.97) ADRB1ADRB2CYP2D6NR3C1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108680676-B Method for quantitatively detecting beta-receptor blocker medicines in dairy products 中国检验检疫科学研究院 2021-08-13 CN claimed
CN-108680676-B Method for quantitatively detecting beta-receptor blocker medicines in dairy products 中国检验检疫科学研究院 2021-08-13 CN disclosed
US-20140088189-A1 METHODS FOR REDUCING THE RISK OF AN ADVERSE DRONEDARONE / BETA-BLOCKERS INTERACTION IN A PATIENT SUFFERING FROM ATRIAL FIBRILATION SANOFI (FR) 2014-03-27 US disclosed
US-8602215-B2 Methods for reducing the risk of an adverse dronedarone/beta-blockers interaction in a patient suffering from atrial fibrillation SANOFI (FR) 2013-12-10 US disclosed
US-20120000806-A1 METHODS FOR REDUCING THE RISK OF AN ADVERSE DRONEDARONE / BETA-BLOCKERS INTERACTION IN A PATIENT SUFFERING FROM ATRIAL FIBRILATION SANOFI (FR) 2012-01-05 US disclosed
WO-2005038049-A2 SYSTEM AND METHOD FOR OPTIMIZING DRUG THERAPY HEINRICH GUENTHER (DE) 2005-04-28 WO disclosed