SCHEMBL5854730

SCHEMBL5854730

COCOc1ccc2c(c1)OCC(C)(c1ccc(O)cc1)C2=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.38
PTPN1 P18031 2/20 0.36
KCNH2 Q12809 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
MAOB P27338 8/20 0.36
MAOA P21397 1/20 0.36
HPGD P15428 3/20 0.34
ALDH1A1 P00352 2/20 0.34
NPC1 O15118 1/20 0.34
NFKB1 P19838 1/20 0.34
GRM5 P41594 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CYP3A4 P08684 2/20 0.34
MAPT P10636 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5854508 0.93 CYP19A1 (0.37) CYP19A1KCNH2TRPV1MAOBMAOA
SCHEMBL5856692 0.86 MAOB (0.52) MAOBMAOAHPGDALDH1A1NPC1
SCHEMBL5855134 0.82 KDM4E (0.46) CYP19A1PTPN1ESR1ESR2MAOB
SCHEMBL5855991 0.80 CYP19A1 (0.47) CYP19A1KCNH2TRPV1MAOBHPGD
SCHEMBL5854453 0.76 CYP19A1 (0.36) CYP19A1KCNH2TRPV1MAOBMAOA
SCHEMBL27560344 0.74 PTPN1 (0.40) CYP19A1PTPN1ESR1ESR2
SCHEMBL5853930 0.73 PTPN1 (0.41) CYP19A1PTPN1ESR1ESR2HPGD
SCHEMBL5855367 0.73 MAOB (0.44) CYP19A1MAOBHPGDALDH1A1SMN1; SMN2
SCHEMBL3357310 0.72 CYP19A1 (0.43) CYP19A1PTPN1ESR1ESR2MAOB
SCHEMBL5854449 0.70 KDM4E (0.36) MAOBMAOAALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7074819-B2 Benzopyran or thiobenzopyran derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2006-07-11 US disclosed
US-20040102479-A1 Novel benzopyran or thiobenzopyran derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA 2004-05-27 US disclosed
US-6645951-B1 Antiestrogens for treating breast cancer CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-11-11 US disclosed
EP-1087959-A1 NOVEL BENZOPYRAN OR THIOBENZOPYRAN DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-04-04 EP disclosed
WO-1999065893-A1 NOVEL BENZOPYRAN OR THIOBENZOPYRAN DERIVATIVES C & C RESEARCH LABORATORIES (KR) 1999-12-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040102479-A1 Novel benzopyran or thiobenzopyran derivatives NR5A1, SHBG, ESR2 CYP19A1 4/4885PTPN1 384/4885KCNH2 3734/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.