SCHEMBL5855112

SCHEMBL5855112

C=CCOCC(OC(=O)C=CC(=O)O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 4/20 0.51
CYP2C19 P33261 1/20 0.38
CYP2D6 P10635 1/20 0.37
CYP3A4 P08684 1/20 0.36
NOS2 P35228 2/20 0.34
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MAPT P10636 2/20 0.33
MDM4 O15151 1/20 0.33
LMNA P02545 1/20 0.33
MDM2 Q00987 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5855848 0.96 HCAR2 (0.44) HCAR2CYP2C19CYP2D6CYP3A4PPARG
SCHEMBL9709425 0.84 HCAR2 (0.58) HCAR2CYP2C19NOS2PPARGPPARA
SCHEMBL9860853 0.84 HCAR2 (0.58) HCAR2CYP2C19NOS2PPARGPPARA
SCHEMBL9709424 0.84 HCAR2 (0.58) HCAR2CYP2C19NOS2PPARGPPARA
SCHEMBL11127289 0.77 CYP2C19 (0.37) CYP2C19CYP2D6CYP3A4PPARGPPARA
SCHEMBL2487162 0.77 HCAR2 (0.59) HCAR2CYP2C19CYP2D6ALDH1A1LMNA
SCHEMBL3482642 0.77 HCAR2 (0.64) HCAR2CYP2C19CYP3A4NOS2ALDH1A1
SCHEMBL3482700 0.77 HCAR2 (0.64) HCAR2CYP2C19CYP3A4NOS2ALDH1A1
SCHEMBL27216283 0.77 HCAR2 (0.64) HCAR2CYP2C19CYP3A4NOS2ALDH1A1
SCHEMBL27741031 0.75 MAPT (0.39) CYP2C19CYP2D6CYP3A4ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7038076-B2 Fumarate derivative, method for producing the same SHOWA DENKO K.K. (JP) 2006-05-02 US disclosed
CN-1181040-C Fumarate derivative and process for producing the same 昭和电工株式会社 2004-12-22 CN disclosed
EP-1301461-A2 FUMARATE DERIVATIVE, METHOD FOR PRODUCING THE SAME Showa Denko K.K. (JP) 2003-04-16 EP disclosed
US-20030060563-A1 Fumarate derivative, method for producing the same SHOWA DENKO K.K. (JP) 2003-03-27 US disclosed
CN-1386116-A Fumarate derivative, method for producing the same SHOWA DENKO KK (JP) 2002-12-18 CN disclosed
WO-2002006206-A2 FUMARATE DERIVATIVE, METHOD FOR PRODUCING THE SAME SHOWA DENKO K.K. (JP) 2002-01-24 WO disclosed