SCHEMBL5855848

SCHEMBL5855848

C=CCOCC(OC(=O)C=CC(=O)OC(COCC=C)c1ccccc1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.44
CYP2C19 P33261 1/20 0.41
CYP2D6 P10635 2/20 0.39
CYP3A4 P08684 2/20 0.38
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
MDM4 O15151 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
MDM2 Q00987 1/20 0.35
ALDH1A1 P00352 3/20 0.34
PKM P14618 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
CYP1A2 P05177 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA7 P43166 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5855112 0.96 HCAR2 (0.51) HCAR2CYP2C19CYP2D6CYP3A4PPARG
SCHEMBL11127289 0.81 CYP2C19 (0.37) CYP2C19CYP2D6CYP3A4PPARGPPARA
SCHEMBL9709424 0.79 HCAR2 (0.58) HCAR2CYP2C19PPARGPPARAMDM4
SCHEMBL9860853 0.79 HCAR2 (0.58) HCAR2CYP2C19PPARGPPARAMDM4
SCHEMBL9709425 0.79 HCAR2 (0.58) HCAR2CYP2C19PPARGPPARAMDM4
SCHEMBL27720282 0.79 MAPT (0.39) CYP2C19CYP2D6CYP3A4LMNAMAPT
SCHEMBL27741031 0.79 MAPT (0.39) CYP2C19CYP2D6CYP3A4LMNAMAPT
SCHEMBL9738617 0.75 THRB (0.40) HCAR2CYP2C19CYP2D6PPARGPPARA
SCHEMBL8067297 0.75 CYP2D6 (0.39) CYP2C19CYP2D6CYP3A4MAPTALDH1A1
SCHEMBL13979422 0.75 CYP2D6 (0.39) CYP2C19CYP2D6CYP3A4MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7038076-B2 Fumarate derivative, method for producing the same SHOWA DENKO K.K. (JP) 2006-05-02 US disclosed
US-20030060563-A1 Fumarate derivative, method for producing the same SHOWA DENKO K.K. (JP) 2003-03-27 US disclosed