SCHEMBL5855973

SCHEMBL5855973

COCOc1ccc(C2(C)COc3cc(OCOC)ccc3C2c2ccc(OCCCCC(CCCC(F)(F)C(F)(F)F)(C(=O)O)C(=O)O)cc2)cc1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.35
PPARD Q03181 16/20 0.35
PPARG P37231 14/20 0.35
FFAR1 O14842 9/20 0.35
PPARA Q07869 3/20 0.33
EDNRB P24530 1/20 0.31
EDNRA P25101 1/20 0.31
CPT1A P50416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5856128 0.91 ESR1 (0.34) ESR1PPARDPPARGFFAR1CPT1A
SCHEMBL5854837 0.90 ESR1 (0.41) ESR1PPARDPPARGFFAR1EDNRB
SCHEMBL5856488 0.83 AR (0.33) PPARDPPARGFFAR1PPARA
SCHEMBL5856257 0.82 FFAR1 (0.31) PPARDPPARGFFAR1
SCHEMBL7587424 0.81 ESR1 (0.32) ESR1PPARDPPARG
SCHEMBL8520859 0.80 PPARG (0.30) ESR1PPARDPPARG
SCHEMBL6938280 0.79 PPARG (0.32) ESR1PPARDPPARGFFAR1EDNRB
SCHEMBL6789008 0.79 ESR1 (0.43) ESR1
SCHEMBL5854374 0.79 PTPN1 (0.35) ESR1PPARDPPARGFFAR1PPARA
SCHEMBL5855606 0.79 ESR1 (0.39) ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7074819-B2 Benzopyran or thiobenzopyran derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2006-07-11 US disclosed
US-6645951-B1 Antiestrogens for treating breast cancer CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-11-11 US disclosed
EP-1087959-A1 NOVEL BENZOPYRAN OR THIOBENZOPYRAN DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-04-04 EP disclosed
WO-1999065893-A1 NOVEL BENZOPYRAN OR THIOBENZOPYRAN DERIVATIVES C & C RESEARCH LABORATORIES (KR) 1999-12-23 WO disclosed