SCHEMBL5864233

SCHEMBL5864233

O=C(O)c1ccc2c(c1)C(=O)N(CCCCCCN1C(=O)c3ccc(C(=O)O)cc3C1=O)C2=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.86
POLB P06746 3/20 0.69
ALDH1A1 P00352 3/20 0.68
TSHR P16473 1/20 0.65
KMT2A Q03164 3/20 0.63
MEN1 O00255 2/20 0.63
HPGD P15428 1/20 0.63
GAA P10253 2/20 0.58
CA1 P00915 2/20 0.58
CA2 P00918 2/20 0.58
CA4 P22748 2/20 0.58
CA9 Q16790 2/20 0.58
ENPP2 Q13822 1/20 0.57
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
HSD17B10 Q99714 2/20 0.54
CASP1 P29466 1/20 0.54
KDM4E B2RXH2 2/20 0.53
MAPK1 P28482 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11033307 0.94 SMN1; SMN2 (0.77) SMN1; SMN2POLBALDH1A1TSHRKMT2A
SCHEMBL9201916 0.94 SMN1; SMN2 (0.77) SMN1; SMN2POLBALDH1A1TSHRKMT2A
SCHEMBL11724761 0.94 SMN1; SMN2 (0.77) SMN1; SMN2POLBALDH1A1TSHRKMT2A
SCHEMBL28350853 0.93 SMN1; SMN2 (0.75) SMN1; SMN2POLBALDH1A1TSHRKMT2A
SCHEMBL28347403 0.93 SMN1; SMN2 (0.75) SMN1; SMN2POLBALDH1A1TSHRKMT2A
SCHEMBL10353400 0.93 SMN1; SMN2 (0.75) SMN1; SMN2POLBALDH1A1TSHRKMT2A
SCHEMBL292284 0.93 SMN1; SMN2 (1.00) SMN1; SMN2POLBALDH1A1TSHRKMT2A
SCHEMBL8344447 0.93 SMN1; SMN2 (0.75) SMN1; SMN2POLBALDH1A1TSHRKMT2A
SCHEMBL17973600 0.93 SMN1; SMN2 (1.00) SMN1; SMN2POLBALDH1A1TSHRKMT2A
SCHEMBL11723011 0.92 SMN1; SMN2 (0.74) SMN1; SMN2POLBALDH1A1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7009027-B2 Graft polymers formed by using polyesterimides having cyclic dicarboxylic anhydride end groups; blends used to form carpet filaments or fibers THUERINGISCHES INSTITUT FUER TEXTIL-UND KUNSTSTOFF-FORSCHUNG E.V. (DE) 2006-03-07 US claimed
EP-1339773-B1 METHOD FOR PRODUCING MELTABLE POLYESTERS THUERINGISCHES INST TEXTIL (DE) 2005-02-02 EP claimed
US-20040039137-A1 Graft polymers formed by using polyesterimides having cyclic dicarboxylic anhydride end groups; blends used to form carpet filaments or fibers THUERINGISCHES INSTITUT FUER TEXTIL-UND KUNSTSTOFF-FORSCHUNG E.V. (DE) 2004-02-26 US claimed
EP-1339773-A2 METHOD FOR PRODUCING MELTABLE POLYESTERS THÜRINGISCHES INSTITUT FÜR TEXTIL- UND KUNSTSTOFF-FORSCHUNG E.V. (DE) 2003-09-03 EP claimed
WO-2002042353-A2 METHOD FOR PRODUCING MELTABLE POLYESTERS THÜRINGISCHES INSTITUT FÜR TEXTIL - UND KUNSTSTOFF - FORSCHUNG E.V. (DE) 2002-05-30 WO claimed
US-7009027-B2 Graft polymers formed by using polyesterimides having cyclic dicarboxylic anhydride end groups; blends used to form carpet filaments or fibers THUERINGISCHES INSTITUT FUER TEXTIL-UND KUNSTSTOFF-FORSCHUNG E.V. (DE) 2006-03-07 US disclosed
EP-1339773-B1 METHOD FOR PRODUCING MELTABLE POLYESTERS THUERINGISCHES INST TEXTIL (DE) 2005-02-02 EP disclosed
US-20040039137-A1 Graft polymers formed by using polyesterimides having cyclic dicarboxylic anhydride end groups; blends used to form carpet filaments or fibers THUERINGISCHES INSTITUT FUER TEXTIL-UND KUNSTSTOFF-FORSCHUNG E.V. (DE) 2004-02-26 US disclosed
EP-1339773-A2 METHOD FOR PRODUCING MELTABLE POLYESTERS THÜRINGISCHES INSTITUT FÜR TEXTIL- UND KUNSTSTOFF-FORSCHUNG E.V. (DE) 2003-09-03 EP disclosed
WO-2002042353-A2 METHOD FOR PRODUCING MELTABLE POLYESTERS THÜRINGISCHES INSTITUT FÜR TEXTIL - UND KUNSTSTOFF - FORSCHUNG E.V. (DE) 2002-05-30 WO disclosed
US-4812377-A CONTAINS 2,3-DIHYDRO-1,3-DIOXO-1H-ISOINDOLE CARBOXYLIC ACIDS EASTMAN KODAK COMPANY (US) 1989-03-14 US disclosed
US-4429108-A HIGH STRENGTH, HEAT RESISTANT FIBERS, FILMS, COATINGS, MOLDINGS STANDARD OIL COMPANY (INDIANA) (US) 1984-01-31 US disclosed
US-3969290-A POLYMERS FROM OXAMIDIC ESTERS, POLYISOCYANATES, AND POLYBASIC CARBOXYLIC ACIDS HOECHST AKTIENGESELLSCHAFT (DT) 1976-07-13 US disclosed