SCHEMBL5864477

SCHEMBL5864477

O=C(CNC(=O)[C@@H]1CCCC[C@H]1c1ccc(Cn2c(CO)nc3ccccc32)cc1)Nc1ccc(F)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.48
LMNA P02545 4/20 0.46
MAPT P10636 4/20 0.46
POLB P06746 2/20 0.43
RAB9A P51151 2/20 0.43
TP53 P04637 3/20 0.42
MCHR1 Q99705 2/20 0.41
CYP2D6 P10635 5/20 0.41
HRH1 P35367 5/20 0.41
CHRM1 P11229 2/20 0.41
GRM2 Q14416 1/20 0.40
KCNH2 Q12809 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5864422 0.94 POLB (0.46) GAALMNAMAPTPOLBRAB9A
SCHEMBL5864345 0.92 POLB (0.44) GAALMNAMAPTPOLBRAB9A
SCHEMBL5864471 0.87 GAA (0.46) GAAPOLBRAB9ATP53MCHR1
SCHEMBL5864499 0.87 POLB (0.45) MAPTPOLBSMN1; SMN2
SCHEMBL5864419 0.81 POLB (0.44) GAALMNAPOLBRAB9ATP53
SCHEMBL5864750 0.80 ALDH1A1 (0.40) POLBTP53ALDH1A1SMN1; SMN2
SCHEMBL5864337 0.80 POLB (0.43) GAAPOLBRAB9ATP53CYP2D6
SCHEMBL5864465 0.79 PDE6D (0.44) GAACYP2D6HRH1CHRM1KCNH2
Hydrochloric Acid SCHEMBL6777163 0.78 PDE6D (0.44) GAAMAPTCYP2D6HRH1CHRM1
SCHEMBL5864495 0.74 HTT (0.40) LMNAPOLBRAB9AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6984642-B1 Substituted phenylcyclohexane carboxylic acid amides and their use as adenosine uptake inhibitors BAYER AKTIENGESELLSCHAFT (DE) 2006-01-10 US disclosed