SCHEMBL5864495

SCHEMBL5864495

O=C(CNC(=O)[C@@H]1CCCC[C@H]1c1ccc(Cn2c(CN3CCOCC3)nc3ncccc32)cc1)Nc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 1/20 0.40
HIF1A Q16665 1/20 0.39
EPAS1 Q99814 1/20 0.39
MOK Q9UQ07 1/20 0.39
BCHE P06276 1/20 0.39
HRH3 Q9Y5N1 2/20 0.39
LMNA P02545 2/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 5/20 0.36
TSHR P16473 1/20 0.36
USP2 O75604 1/20 0.36
HPGD P15428 1/20 0.36
P2RX3 P56373 1/20 0.36
AVPR1A P37288 1/20 0.36
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5864489 0.85 CYP1A2 (0.40) HIF1ALMNAKMT2AALDH1A1TSHR
SCHEMBL5864492 0.81 KDM4E (0.38) MOKBCHEALDH1A1TSHRAVPR1A
SCHEMBL6214082 0.79 GRM2 (0.39) SMN1; SMN2NPC1RAB9AHIF1ALMNA
SCHEMBL5864499 0.78 POLB (0.45) SMN1; SMN2POLB
Hydrochloric Acid SCHEMBL6779410 0.78 ULK1 (0.40) HTTSMN1; SMN2NPC1RAB9AMOK
SCHEMBL5864465 0.75 PDE6D (0.44)
Hydrochloric Acid SCHEMBL6777163 0.74 PDE6D (0.44) KMT2AALDH1A1TSHR
SCHEMBL5864477 0.74 GAA (0.48) SMN1; SMN2RAB9ALMNAPOLBKMT2A
SCHEMBL5864750 0.73 ALDH1A1 (0.40) SMN1; SMN2POLBALDH1A1
SCHEMBL5864422 0.73 POLB (0.46) RAB9ALMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6984642-B1 Substituted phenylcyclohexane carboxylic acid amides and their use as adenosine uptake inhibitors BAYER AKTIENGESELLSCHAFT (DE) 2006-01-10 US disclosed
EP-1187812-B1 SUBSTITUTED PHENYLCYCLOHEXANE CARBOXYLIC ACID AMIDES AND THEIR USE AS ADENOSINE UPTAKE INHIBITORS BAYER HEALTHCARE AG (DE) 2005-09-07 EP disclosed
US-6716849-B1 ISCHEMIC BRAIN DISORDERS; NEUROPROTECTANTS BAYER AKTIENGESELLSCHAFT (DE) 2004-04-06 US disclosed