SCHEMBL5865098

SCHEMBL5865098

CCOC(=O)CS(=O)(=O)Nc1ccc(OC2CCN(C)CC2)c(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.46
BRAF P15056 3/20 0.46
KDR P35968 2/20 0.46
F2 P00734 5/20 0.45
F10 P00742 5/20 0.45
UTS2R Q9UKP6 3/20 0.44
BRD4 O60885 2/20 0.44
RAF1 P04049 2/20 0.43
ARAF P10398 2/20 0.43
ABL1 P00519 1/20 0.43
MAPK14 Q16539 1/20 0.42
FGFR1 P11362 1/20 0.42
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
FPR2 P25090 2/20 0.41
PROKR1 Q8TCW9 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5865273 0.88 GPR119 (0.49) RORCBRD4
SCHEMBL5864995 0.88 RORC (0.49) RORCUTS2RBRD4KDM4ELMNA
SCHEMBL5865064 0.79 RORC (0.48) RORCUTS2RKDM4ELMNAFPR2
SCHEMBL21465789 0.79 BRAF (0.57) RORCBRAFKDRF2F10
SCHEMBL5864927 0.79 RORC (0.50) RORCKDM4ELMNAMAPTNPSR1
SCHEMBL5864987 0.79 SMN1; SMN2 (0.49) RORCLMNAFPR2PROKR1
SCHEMBL5864923 0.78 RORC (0.45) RORCKDM4ELMNA
SCHEMBL5865205 0.78 RORC (0.47) RORCF2F10KDM4ELMNA
SCHEMBL5864758 0.78 RORC (0.47) RORC
SCHEMBL5864754 0.77 KDM4E (0.49) RORCKDM4ELMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7030138-B2 Benzamidine derivatives SANKYO COMPANY, LIMITED (JP) 2006-04-18 US disclosed
US-20040147555-A1 Benzamidine derivatives SANKYO COMPANY, LIMITED (JP) 2004-07-29 US disclosed
EP-1375482-A1 BENZAMIDINE DERIVATIVE Sankyo Company, Limited (JP) 2004-01-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040147555-A1 Benzamidine derivatives F9, F7, F2 RORC 4836/4885BRAF 228/4885KDR 1062/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.