SCHEMBL586551

SCHEMBL586551

CC1(C)OB(c2ccc(OC(F)(F)F)cc2F)OC1(C)C.Fc1cc(OC(F)(F)F)ccc1Br

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 1/20 0.39
LIPE Q05469 4/20 0.37
PDE2A O00408 1/20 0.34
GPR3 P46089 4/20 0.33
GRM2 Q14416 1/20 0.32
CCR6 P51684 1/20 0.31
LPL P06858 1/20 0.31
LIPG Q9Y5X9 1/20 0.31
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
GAA P10253 1/20 0.30
THRB P10828 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30
CES1 P23141 1/20 0.30
SLC6A4 P31645 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL581309 0.92 CXCR2 (0.43) CXCR2LIPEPDE2AGPR3GRM2
SCHEMBL30376702 0.92 CXCR2 (0.43) CXCR2LIPEPDE2AGPR3GRM2
SCHEMBL14874698 0.85 SNCA (0.37) LPLLIPGCA1CA2CA9
SCHEMBL17129378 0.79 AR (0.42) CXCR2LIPEALDH1A1
SCHEMBL30377217 0.78 GPR3 (0.46) PDE2AGPR3ALDH1A1POLBGAA
SCHEMBL518353 0.78 GPR3 (0.46) PDE2AGPR3ALDH1A1POLBGAA
SCHEMBL15572934 0.78 PTGS1 (0.38)
SCHEMBL15573245 0.78 ALK (0.32)
SCHEMBL20191122 0.78 CXCR2 (0.41) CXCR2LIPEGPR3CA1CA2
SCHEMBL28961843 0.77 CXCR2 (0.42) CXCR2LIPEGPR3CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed