SCHEMBL5865840

SCHEMBL5865840

Cn1c(=O)cc(C(F)(F)F)c2cc(S(=O)(=O)N3CCCC4CCCC=C43)ccc21

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AR P10275 16/20 0.40
PGR P06401 5/20 0.40
NR3C1 P04150 1/20 0.40
NR3C2 P08235 1/20 0.40
KDM4E B2RXH2 1/20 0.37
USP2 O75604 2/20 0.37
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PARG Q86W56 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5865913 0.82 AR (0.49) ARPGRNR3C1NR3C2KDM4E
SCHEMBL5865841 0.76 AR (0.46) ARPGRNR3C1NR3C2KDM4E
SCHEMBL5865914 0.76 HSD17B10 (0.57) ARKDM4EUSP2ALDH1A1HPGD
SCHEMBL5865901 0.76 HSD17B10 (0.57) ARKDM4EUSP2ALDH1A1HPGD
SCHEMBL5865876 0.74 ALDH1A1 (0.64) ALDH1A1TSHR
SCHEMBL6106171 0.73 AR (0.44) AR
SCHEMBL6022453 0.73 AR (0.48) ARPGRNR3C1NR3C2USP2
SCHEMBL6105325 0.72 MAOB (0.37) ARPGRKDM4EUSP2ALDH1A1
SCHEMBL5865896 0.72 AR (0.47) ARPGRNR3C1NR3C2USP2
SCHEMBL6023005 0.70 PIK3CG (0.57) ARPGRNR3C1NR3C2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7064207-B2 6-sulfonamido-quinolin-2-one and 6-sulfonamido-2-oxo-chromene derivatives, useful for treating alopecia, acne and oily skin WARNER LAMBERT COMPANY LLC (US) 2006-06-20 US claimed
US-20050085467-A1 Androgen receptor antagonists DU DANIEL Y (US) 2005-04-21 US claimed
US-7064207-B2 6-sulfonamido-quinolin-2-one and 6-sulfonamido-2-oxo-chromene derivatives, useful for treating alopecia, acne and oily skin WARNER LAMBERT COMPANY LLC (US) 2006-06-20 US disclosed
EP-1587804-A1 ANDROGEN RECEPTOR ANTAGONISTS Warner-Lambert Company LLC (US) 2005-10-26 EP disclosed
US-20050085467-A1 Androgen receptor antagonists DU DANIEL Y (US) 2005-04-21 US disclosed
WO-2004065379-A1 ANDROGEN RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY LLC (US) 2004-08-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050085467-A1 Androgen receptor antagonists AR, NR5A1, ESRRB AR 1/4885PGR 100/4885NR3C1 44/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.