SCHEMBL5866414

SCHEMBL5866414

[CH2]C(CCN1CCC(N2CCCN(CC(=O)NC)C2=O)CC1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.61

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 16/20 0.61
TACR1 P25103 16/20 0.61
TACR3 P29371 16/20 0.61
MCHR1 Q99705 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5866449 0.87 TACR2 (0.49) TACR2TACR1TACR3MCHR1
Citric Acid SCHEMBL7044834 0.76 TACR2 (0.58) TACR2TACR1TACR3
SCHEMBL5866420 0.75 TACR2 (0.48) TACR2TACR1TACR3MCHR1
SCHEMBL5866423 0.73 TACR2 (0.61) TACR2
SCHEMBL8314527 0.72 HDAC1 (0.45) TACR2MCHR1
Citric Acid SCHEMBL5866407 0.71 TACR2 (0.43) TACR2TACR1TACR3MCHR1
SCHEMBL1387917 0.70 TACR2 (0.70) TACR2
SCHEMBL1387915 0.70 TACR2 (0.70) TACR2
SCHEMBL6959139 0.70 CCR5 (0.57) TACR2TACR1TACR3
SCHEMBL6963702 0.69 CCR5 (0.50) TACR2MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7053213-B2 Therapeutic heterocycles ASTRAZENECA AB (SE) 2006-05-30 US claimed
US-7053213-B2 Therapeutic heterocycles ASTRAZENECA AB (SE) 2006-05-30 US disclosed
EP-0714392-B1 HETEROCYCLES USEFUL AS NEUROKININ ANTAGONISTS ZENECA LTD (GB) 1998-11-04 EP disclosed