SCHEMBL5869592

SCHEMBL5869592

COC(=O)[C@@H](N)Cc1cc(-c2ccccc2)on1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.52
CYP1A2 P05177 2/20 0.50
CYP2D6 P10635 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
STAT3 P40763 1/20 0.48
STAT1 P42224 1/20 0.48
RAB9A P51151 4/20 0.48
ALDH1A1 P00352 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
MAPT P10636 2/20 0.47
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5869598 1.00 NOTUM (0.52) NOTUMCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL1118444 0.79 F10 (0.47)
SCHEMBL1118442 0.79 F10 (0.47)
SCHEMBL6499726 0.78 KDM4E (0.55) RAB9AALDH1A1SMN1; SMN2L3MBTL1MAPT
SCHEMBL8296884 0.78 KDM4E (0.55) RAB9AALDH1A1SMN1; SMN2L3MBTL1MAPT
SCHEMBL12002394 0.78 NOTUM (0.58) NOTUMCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL14210011 0.77 NOTUM (0.65) NOTUMCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6809054 0.75 NOTUM (0.51) NOTUMRAB9AALDH1A1SMN1; SMN2MAPT
Phenylalanine Methyl Ester SCHEMBL27535118 0.74 SLC7A5 (0.58) CYP2C9CYP2C19ALDH1A1POLBKMT2A
SCHEMBL14552880 0.74 RAB9A (0.67) NOTUMRAB9AALDH1A1SMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7045532-B2 ACE-2 modulating compounds and methods of use thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2006-05-16 US disclosed
US-20040082496-A1 ACE-2 modulating compounds and methods of use thereof MILLENNIUM PHARMACEUTICALS, INC. 2004-04-29 US disclosed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040082496-A1 ACE-2 modulating compounds and methods of use thereof ACE, ACE2, AGTR2 NOTUM 1226/4885CYP1A2 827/4885CYP2D6 607/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.