SCHEMBL587170

SCHEMBL587170

CCOC(=O)CC(=O)C1CCN(C(=O)O)C(c2nnnn2C)C1.Cn1nnnc1C1CC(C(=O)O)CCN1C(=O)OCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 9/20 0.42
TMEM97 Q5BJF2 8/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL587119 0.95 SIGMAR1 (0.45) SIGMAR1TMEM97NPC1RAB9ASMN1; SMN2
SCHEMBL587171 0.91 SIGMAR1 (0.42) SIGMAR1TMEM97NPC1RAB9AALDH1A1
SCHEMBL586903 0.88 SMN1; SMN2 (0.51) SIGMAR1TMEM97NPC1RAB9ASMN1; SMN2
SCHEMBL587054 0.87 MAPK1 (0.36) NPC1RAB9AALDH1A1
SCHEMBL586922 0.85 ALDH1A1 (0.49) SIGMAR1TMEM97NPC1RAB9ASMN1; SMN2
SCHEMBL586771 0.83 SIGMAR1 (0.43) SIGMAR1TMEM97NPC1RAB9ASMN1; SMN2
SCHEMBL582341 0.80 SIGMAR1 (0.45) SIGMAR1TMEM97HTT
SCHEMBL2991986 0.76 TMEM97 (0.51) SIGMAR1TMEM97
SCHEMBL2991989 0.76 TMEM97 (0.51) SIGMAR1TMEM97
SCHEMBL586708 0.75 ALDH1A1 (0.42) NPC1RAB9ASMN1; SMN2ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed