SCHEMBL5872919

SCHEMBL5872919

Cc1cc(I)ccc1Nc1c(C(=O)O)cc(C(=O)NCCCN2CCCC2=O)c(F)c1F

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.46
USP2 O75604 1/20 0.45
RECQL P46063 1/20 0.45
FSHR P23945 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 2/20 0.44
GAA P10253 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5872920 0.97 RAB9A (0.49) RAB9AL3MBTL1USP2RECQLFSHR
SCHEMBL5872857 0.83 BCL3 (0.48) L3MBTL1SMN1; SMN2KMT2AALDH1A1KDM4E
SCHEMBL5872926 0.80 MEN1 (0.47) KMT2A
SCHEMBL5872804 0.80 BCL3 (0.47) KMT2AALDH1A1LMNA
SCHEMBL5872816 0.79 MEN1 (0.50) SMN1; SMN2KMT2AALDH1A1KDM4EHPGD
SCHEMBL5872844 0.79 KMT2A (0.47) SMN1; SMN2KMT2AALDH1A1KDM4E
SCHEMBL5872928 0.77 MEN1 (0.49) KMT2A
SCHEMBL5872807 0.76 MEN1 (0.48) KMT2AALDH1A1LMNA
SCHEMBL5872818 0.76 MEN1 (0.50) SMN1; SMN2KMT2AALDH1A1KDM4EHPGD
SCHEMBL5872850 0.76 MAP2K1 (0.56) SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7001905-B2 Substituted diarylamines as MEK inhibitors WARNER-LAMBERT COMPANY (US) 2006-02-21 US disclosed
US-20030225076-A1 5-Amide substituted diarylamines as mex inhibitors BIWERSI CATHLIN (US) 2003-12-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030225076-A1 5-Amide substituted diarylamines as mex inhibitors NRAS, MAPK6, MAPK12 RAB9A 3021/4885L3MBTL1 2631/4885USP2 4601/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.