SCHEMBL5873084

SCHEMBL5873084

COC(=O)[C@@H](C)CO[Si](c1ccccc1)(c1ccccc1)C(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ESRRB O95718 1/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 2/20 0.37
THRB P10828 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HSD17B10 Q99714 1/20 0.37
HPGD P15428 1/20 0.37
MAPT P10636 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
CYP3A4 P08684 1/20 0.36
HTT P42858 1/20 0.36
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36
ABL1 P00519 1/20 0.36
SMYD2 Q9NRG4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5685150 1.00 ESRRB (0.39) ESRRBKMT2AALDH1A1THRBCYP2C9
SCHEMBL5685142 1.00 ESRRB (0.39) ESRRBKMT2AALDH1A1THRBCYP2C9
SCHEMBL4706102 0.87 APAF1 (0.37) ALDH1A1CYP2C19SMN1; SMN2CYP3A4HTT
SCHEMBL4706098 0.87 APAF1 (0.37) ALDH1A1CYP2C19SMN1; SMN2CYP3A4HTT
SCHEMBL451543 0.87 APAF1 (0.37) ALDH1A1CYP2C19SMN1; SMN2CYP3A4HTT
Hydrochloric Acid SCHEMBL4708235 0.87 APAF1 (0.37) ALDH1A1CYP2C19SMN1; SMN2CYP3A4HTT
Hydrochloric Acid SCHEMBL4708232 0.87 APAF1 (0.37) ALDH1A1CYP2C19SMN1; SMN2CYP3A4HTT
SCHEMBL7898284 0.86 KMT2A (0.39) KMT2AALDH1A1MAPTL3MBTL1SMN1; SMN2
SCHEMBL6633064 0.85 CYP3A4 (0.35) ALDH1A1HPGDSMN1; SMN2CYP3A4HTT
SCHEMBL6636609 0.85 CYP3A4 (0.35) ALDH1A1HPGDSMN1; SMN2CYP3A4HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024129763-A1 MODULATORS OF TNF-α ACTIVITY FORWARD THERAPEUTICS, INC. (US) 2024-06-20 WO disclosed
CN-114644627-B AhR inhibitors and uses thereof 山东轩竹医药科技有限公司 2024-06-11 CN disclosed
CN-115698005-B Fused ring AhR inhibitors 山东轩竹医药科技有限公司 2024-02-06 CN disclosed
WO-2022127753-A1 FUSED RING AHR INHIBITOR 山东轩竹医药科技有限公司 2022-06-23 WO disclosed
CN-114644627-A AhR inhibitor and application thereof 山东轩竹医药科技有限公司 2022-06-21 CN disclosed
US-6982257-B1 Vitamin D3 derivative and its production method TEIJIN LIMITED (JP) 2006-01-03 US disclosed