SCHEMBL5873731

SCHEMBL5873731

C=CN1C(=O)Cc2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.50
NOTUM Q6P988 1/20 0.47
DDB1 Q16531 1/20 0.40
CRBN Q96SW2 1/20 0.40
KMT2A Q03164 2/20 0.39
CASP3 P42574 1/20 0.39
CASP6 P55212 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
OPRM1 P35372 4/20 0.39
OPRK1 P41145 4/20 0.39
OPRL1 P41146 4/20 0.39
HTR7 P34969 4/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
RNASEH1 O60930 1/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31726238 1.00 HPGD (0.50) HPGDNOTUMDDB1CRBNKMT2A
SCHEMBL21457751 0.84 HPGD (0.38) HPGDNOTUMKMT2AOPRM1OPRK1
SCHEMBL4409235 0.82 HPGD (0.56) HPGDNOTUMDDB1CRBNKMT2A
SCHEMBL24049835 0.78 HPGD (0.35) HPGDNOTUMKMT2AOPRM1OPRK1
SCHEMBL318501 0.77 NOTUM (0.47) HPGDNOTUMDDB1CRBNKMT2A
SCHEMBL28669819 0.75 HPGD (0.49) HPGDNOTUMDDB1CRBNKMT2A
SCHEMBL6362724 0.74 KMT2A (0.33) HPGDNOTUMKMT2AMEN1MAPT
SCHEMBL5323856 0.74 HPGD (0.55) HPGDNOTUMDDB1CRBNKMT2A
SCHEMBL30215698 0.73 HTR7 (0.50) HPGDNOTUMCASP3HTR7HTR1A
SCHEMBL185755 0.73 HTR7 (0.50) HPGDNOTUMCASP3HTR7HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111704571-A Preparation method of optically active 2-aryl spiro [ cyclopentane-1, 3' -indole ] -3-formaldehyde 南宁师范大学 2020-09-25 CN claimed
CN-111704571-A Preparation method of optically active 2-aryl spiro [ cyclopentane-1, 3' -indole ] -3-formaldehyde 南宁师范大学 2020-09-25 CN disclosed
CN-111704571-A Preparation method of optically active 2-aryl spiro [ cyclopentane-1, 3' -indole ] -3-formaldehyde 南宁师范大学 2020-09-25 CN disclosed
EP-1317013-B1 NON-AQUEOUS ELECTROLYTE AND SECONDARY CELL USING THE SAME MITSUBISHI CHEM CORP (JP) 2017-03-15 EP disclosed
US-7129253-B2 Compounds SMITHKLINE BEECHAM CORPORATION (US) 2006-10-31 US disclosed
US-6942948-B2 Nonaqueous electrolyte solution and secondary battery employing the same MITSUBISHI CHEMICAL CORPORATION (JP) 2005-09-13 US disclosed
US-20030165733-A1 Nonaqueous electrolyte solution and secondary battery employing the same MITSUBISHI CHEMICAL CORPORATION (JP) 2003-09-04 US disclosed
EP-1317013-A1 NON-AQUEOUS ELECTROLYTE AND SECONDARY CELL USING THE SAME MITSUBISHI CHEMICAL CORPORATION (JP) 2003-06-04 EP disclosed
US-6498176-B1 INHIBITING TUMOR GROWTH VIA INHIBITION OF TUMOR-RELATED ANGIOGENESIS SMITHKLINEBEECHAM CORPORATION 2002-12-24 US disclosed
US-6358750-B1 FOR COMBINATORIAL LIBRARIES; DRUG SCREENING ARQULE, INC. 2002-03-19 US disclosed
EP-1125937-A2 Spiro [Pyrrolidine-2,3'-oxindole] compounds and methods of use ARQULE, INC. (US) 2001-08-22 EP disclosed
EP-1015430-A4 SPIRO PYRROLIDINE-2,3'-OXINDOLE] COMPOUNDS AND METHODS OF USE ARQULE INC (US) 2001-01-17 EP disclosed
US-6114540-A COMBINATORIAL LIBRARIES ARQULE, INC. (US) 2000-09-05 US disclosed
EP-1015430-A1 SPIRO PYRROLIDINE-2,3'-OXINDOLE] COMPOUNDS AND METHODS OF USE ARQULE, INC. (US) 2000-07-05 EP disclosed
WO-1999012904-A1 SPIRO[PYRROLIDINE-2,3'-OXINDOLE] COMPOUNDS AND METHODS OF USE ARQULE, INC. (US) 1999-03-18 WO disclosed