SCHEMBL587855

SCHEMBL587855

CCOC(=O)C1CCN(C(=O)O)C(c2nnn[nH]2)C1.CCOC(=O)C1CCN(C(=O)OCc2ccccc2)C(C#N)C1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 3/20 0.39
SIGMAR1 Q99720 3/20 0.39
ALDH1A1 P00352 2/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
PKM P14618 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PREP P48147 2/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ELANE P08246 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL586528 0.90 TMEM97 (0.46) TMEM97SIGMAR1ALDH1A1NPC1RAB9A
SCHEMBL587386 0.85 PKM (0.48) NPC1RAB9APKMNPSR1PREP
SCHEMBL587226 0.82 POLB (0.39) ALDH1A1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL15878549 0.75 SMN1; SMN2 (0.60) NPC1RAB9APREPSMN1; SMN2
SCHEMBL13103714 0.74 ALDH1A1 (0.35) ALDH1A1NPC1RAB9AMAPT
SCHEMBL586922 0.73 ALDH1A1 (0.49) TMEM97SIGMAR1ALDH1A1NPC1RAB9A
SCHEMBL615936 0.72 CYP3A4 (0.45) ALDH1A1NPC1RAB9APKMNPSR1
SCHEMBL13246605 0.72 TMEM97 (0.49) TMEM97SIGMAR1NPC1RAB9ANPSR1
SCHEMBL672317 0.72 TMEM97 (0.49) TMEM97SIGMAR1NPC1RAB9ANPSR1
SCHEMBL4521587 0.72 TMEM97 (0.49) TMEM97SIGMAR1NPC1RAB9ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed