SCHEMBL5879290

SCHEMBL5879290

C=CCC(C(=O)Cl)c1ccc(Br)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.51
KMT2A Q03164 1/20 0.42
CYP1A2 P05177 1/20 0.42
FFAR2 O15552 1/20 0.40
TGM2 P21980 2/20 0.38
LMNA P02545 2/20 0.37
F13A1 P00488 1/20 0.37
TGM1 P22735 1/20 0.37
TGM3 Q08188 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.35
ALOX5 P09917 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
HTT P42858 1/20 0.34
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13946462 0.86 FFAR2 (0.52) CYP2C19KMT2ACYP1A2FFAR2LMNA
SCHEMBL4264360 0.84 CYP2C19 (0.50) CYP2C19KMT2AFFAR2TGM2LMNA
SCHEMBL6002239 0.84 CYP2C19 (0.50) CYP2C19KMT2AFFAR2TGM2LMNA
SCHEMBL6423644 0.84 CYP2C19 (0.73) CYP2C19FFAR2LMNASMN1; SMN2
SCHEMBL6423647 0.84 CYP2C19 (0.73) CYP2C19FFAR2LMNASMN1; SMN2
SCHEMBL5879152 0.84 CYP2C19 (0.73) CYP2C19KMT2ACYP1A2FFAR2TGM2
SCHEMBL7268439 0.81 CYP2C19 (0.50) CYP2C19KMT2ACYP1A2LMNASMN1; SMN2
SCHEMBL623726 0.78 SLC6A2 (0.44) CYP2C19CYP1A2FFAR2LMNASMN1; SMN2
SCHEMBL5879182 0.78 SLC6A2 (0.44) CYP2C19CYP1A2FFAR2LMNASMN1; SMN2
SCHEMBL5879184 0.78 SLC6A2 (0.44) CYP2C19CYP1A2FFAR2LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7034056-B2 Aryl and biaryl compounds having MCH modulatory activity PHARMACOPEIA DRUG DISCOVERY, INC. (US) 2006-04-25 US disclosed
EP-1370520-A1 ARYL AND BIARYL COMPOUNDS HAVING MCH MODULATORY ACTIVITY PHARMACOPEIA, INC. (US) 2003-12-17 EP disclosed
WO-2002076929-A1 ARYL AND BIARYL COMPOUNDS HAVING MCH MODULATORY ACTIVITY PHARMACOPEIA, INC. (US) 2002-10-03 WO disclosed