SCHEMBL5884420

SCHEMBL5884420

Nc1ccc2cccc(OCC3CCCCC3)c2n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 17/20 1.00
NCF1 P14598 3/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5883835 0.99 MCHR1 (1.00) MCHR1NCF1
SCHEMBL5883878 0.96 MCHR1 (1.00) MCHR1NCF1
SCHEMBL5884166 0.86 MCHR1 (1.00) MCHR1NCF1
SCHEMBL7261142 0.85 MCHR1 (0.88) MCHR1NCF1
SCHEMBL5883858 0.82 MCHR1 (1.00) MCHR1NCF1
SCHEMBL2483278 0.81 MCHR1 (0.68) MCHR1
SCHEMBL5884150 0.79 MCHR1 (1.00) MCHR1NCF1
SCHEMBL28195001 0.78 MCHR1 (0.66) MCHR1NCF1
SCHEMBL5884483 0.78 MCHR1 (1.00) MCHR1NCF1
SCHEMBL5883787 0.78 MCHR1 (1.00) MCHR1NCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6989392-B2 2-Aminoquinolines as melanin concentrating hormone receptor antagonists ABBOTT LABORATORIES (US) 2006-01-24 US claimed
US-20040063756-A1 2-Aminoquinolines as melanin concentrating hormone receptor antagonists ABBVIE INC. 2004-04-01 US claimed
EP-3558298-B1 ANTIDIABETIC SPIROCHROMAN COMPOUNDS MERCK SHARP & DOHME LLC (US) 2026-03-11 EP disclosed
US-20250346646-A1 COMPOUNDS USEFUL TO TREAT METABOLIC DISORDERS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2025-11-13 US disclosed
EP-2958562-B1 ANTIDIABETIC BICYCLIC COMPOUNDS MERCK SHARP & DOHME LLC (US) 2025-09-10 EP disclosed
WO-2024155618-A1 COMPOSITIONS AND METHODS FOR TREATING WEIGHT GAIN AND/OR DISORDERS ASSOCIATED WITH ABNORMAL DE NOVO LIPOGENESIS, AND FAT ACCUMULATION CASE WESTERN RESERVE UNIVERSITY (US) 2024-07-25 WO disclosed
EP-3436003-B1 ANTIDIABETIC BICYCLIC COMPOUNDS MERCK SHARP & DOHME LLC (US) 2023-08-23 EP disclosed
US-20220411490-A1 METHOD TO IDENTIFY COMPOUNDS USEFUL TO TREAT DYSREGULATED LIPOGENESIS, DIABETES, AND RELATED DISORDERS PRESIDENT AND FELLOWS OF HARVARD COLLEGE 2022-12-29 US disclosed
CN-109642908-B Compounds useful for treating metabolic disorders 哈佛学院院长及董事 2022-08-16 CN disclosed
US-11345748-B2 Method of treating idiopathic pulmonary fibrosis and kidney fibrosis PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2022-05-31 US disclosed
US-6989392-B2 2-Aminoquinolines as melanin concentrating hormone receptor antagonists ABBOTT LABORATORIES (US) 2006-01-24 US disclosed
US-20040063756-A1 2-Aminoquinolines as melanin concentrating hormone receptor antagonists ABBVIE INC. 2004-04-01 US disclosed
WO-2003105850-A1 2-AMINOQUINOLINES AS MELANIN CONCENTRATING HORMONE RECEPTOR ANTAGONISTS ABBOTT LABORATORIES (US) 2003-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063756-A1 2-Aminoquinolines as melanin concentrating hormone receptor antagonists MCHR1, MCHR2, MC1R MCHR1 1/4885NCF1 3219/4885
US-11345748-B2 Method of treating idiopathic pulmonary fibrosis and kidney fibrosis CNR2, FABP1, FABP4 MCHR1 1809/4885NCF1 1197/4885
US-20220411490-A1 METHOD TO IDENTIFY COMPOUNDS USEFUL TO TREAT DYSREGULATED LIPOGENESIS, DIABETES, AND RELATED DISORDERS FABP4, LIPC, CNR2 MCHR1 1571/4885NCF1 1835/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.