SCHEMBL5885013

SCHEMBL5885013

COc1cccc(C2=C(c3ccccc3CN(C)C)CCCC2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.50
GRM5 P41594 1/20 0.47
ESR1 P03372 1/20 0.44
ESR2 Q92731 1/20 0.44
PTGER1 P34995 1/20 0.43
HTR7 P34969 3/20 0.41
SLC6A2 P23975 4/20 0.41
SLC6A4 P31645 4/20 0.41
SLC6A3 Q01959 4/20 0.41
HTR1A P08908 1/20 0.40
ABCB1 P08183 1/20 0.40
ABCC1 P33527 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
CYP1A2 P05177 3/20 0.39
CYP3A4 P08684 3/20 0.39
CYP2D6 P10635 3/20 0.39
MAPT P10636 1/20 0.39
MEN1 O00255 1/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6048529 0.84 BACE1 (0.58) BACE1GRM5HTR7SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL6048554 0.83 BACE1 (0.57) BACE1GRM5HTR7SLC6A2SLC6A4
SCHEMBL5884334 0.81 CALM1 (0.42) BACE1GRM5HTR7SLC6A2SLC6A4
SCHEMBL7752297 0.80 MAOB (0.41) GRM5ESR1ESR2HTR7HTR1A
SCHEMBL6680825 0.73 BRD4 (0.49) GRM5ESR1ESR2KDM4E
SCHEMBL6048510 0.70 HTR2A (0.56) BACE1HTR7SLC6A4HTR1AABCB1
SCHEMBL12054106 0.70 CALM1 (0.48) SLC6A2SLC6A4SLC6A3HTR1ATSHR
SCHEMBL6048547 0.69 BACE1 (0.55) BACE1PTGER1HTR7SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL6048492 0.69 HTR2A (0.55) BACE1HTR7SLC6A4HTR1AABCB1
SCHEMBL13007829 0.69 MAOB (0.50) MAPTMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7064236-B2 Substituted 1-aryl-but-3-enylamine and 1-aryl-but-2-enylamine compounds GRUNENTHAL GMBH (DE) 2006-06-20 US claimed