SCHEMBL5886910

SCHEMBL5886910

CC1=C(c2ccc(O)cc2)[CH]CC=C1c1ccc(Cl)c(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.38
AHR P35869 3/20 0.36
ALOX5 P09917 2/20 0.36
VCP P55072 1/20 0.36
ESR2 Q92731 3/20 0.36
ESR1 P03372 2/20 0.36
EGFR P00533 1/20 0.33
ERBB2 P04626 1/20 0.33
CYP1B1 Q16678 1/20 0.33
SRC P12931 1/20 0.32
SLC6A3 Q01959 2/20 0.32
KMO O15229 1/20 0.31
MEN1 O00255 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887415 0.82 AHR (0.38) AHREGFRCYP1B1SLC6A3MEN1
SCHEMBL5886907 0.80 BCL2L1 (0.36) SLC6A3MEN1KMT2A
SCHEMBL4009121 0.71 ALDH1A1 (0.33) MEN1KMT2A
SCHEMBL5887212 0.71 ALKBH3 (0.39) HSD17B10AHREGFRCYP1B1SLC6A3
SCHEMBL5887298 0.70 RAD51 (0.40) AHREGFRSRC
SCHEMBL5887524 0.69 RAD51 (0.37) AHREGFRSRC
SCHEMBL5887017 0.69 EGFR (0.38) AHREGFRCYP1B1SLC6A3
SCHEMBL5887338 0.69 EGFR (0.41) AHREGFRSRC
SCHEMBL6335821 0.68 AHR (0.70) HSD17B10AHRALOX5ESR2ESR1
SCHEMBL5887318 0.68 BCL2L1 (0.37) AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037931-B2 Corticotropin releasing factor moderator; analgesics; drug abruse, drug dependency; schizophrenia JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-02 US disclosed
US-20050020565-A1 Pyrazole compound; gastrointestinal disorders; central nervous system disorders JONES TODD K (US) 2005-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050020565-A1 Pyrazole compound; gastrointestinal disorders; central nervous system disorders CCKAR, CCKBR, NPY1R HSD17B10 1195/4885AHR 16/4885ALOX5 2648/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.