SCHEMBL5887004

SCHEMBL5887004

Cc1nc(N2CCC(C(=O)c3ccc(F)cc3)CC2)nc2c1ccc(=O)n2-c1ccc(C(=O)NC2CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 11/20 0.47
CDK2 P24941 11/20 0.47
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
PAK1 Q13153 1/20 0.40
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40
CCND3 P30281 1/20 0.40
CDK7 P50613 1/20 0.40
CCNH P51946 1/20 0.40
MNAT1 P51948 1/20 0.40
CDK6 Q00534 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
PRKAB2 O43741 1/20 0.40
PRKAG1 P54619 1/20 0.40
PRKAA2 P54646 1/20 0.40
PRKAA1 Q13131 1/20 0.40
PRKAG3 Q9UGI9 1/20 0.40
PRKAG2 Q9UGJ0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887152 0.91 CCNE1 (0.48) CCNE1CDK2CNR1CNR2PAK1
SCHEMBL5887545 0.88 HSD11B1 (0.40) POLB
SCHEMBL5886823 0.87 SMYD3 (0.48) CCNE1CDK2POLB
SCHEMBL5887117 0.86 SMN1; SMN2 (0.49) POLB
SCHEMBL5887242 0.85 BRD4 (0.47) CCNE1CDK2MAPK14
SCHEMBL5887369 0.84 KDM4E (0.41) CCNE1CDK2ALDH1A1
SCHEMBL5887102 0.84 ALDH1A1 (0.40) CCNE1CDK2PAK1ALDH1A1
SCHEMBL5886731 0.84 KDM4E (0.41) POLB
SCHEMBL5887260 0.84 KMT2A (0.42) POLB
SCHEMBL5886718 0.84 CCNE1 (0.45) CCNE1CDK2PDE4BPDE4DMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US claimed
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US disclosed