SCHEMBL5887252

SCHEMBL5887252

Cc1nc(Oc2ccc(C(=O)O)cc2)nc2c1ccc(=O)n2-c1ccc(C(N)=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 4/20 0.45
PARP15 Q460N3 2/20 0.45
RXRA P19793 1/20 0.44
CSNK2A1 P68400 5/20 0.42
MAPK1 P28482 2/20 0.38
ALDH1A1 P00352 8/20 0.38
CYP1A2 P05177 6/20 0.38
CYP3A4 P08684 6/20 0.38
USP2 O75604 5/20 0.38
CLK4 Q9HAZ1 1/20 0.38
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
CYP2C19 P33261 2/20 0.38
TSHR P16473 1/20 0.38
CYP2C9 P11712 3/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP2D6 P10635 1/20 0.37
PARP14 Q460N5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5886767 0.92 ALDH1A1 (0.38) PARP10PARP15RXRACSNK2A1MAPK1
SCHEMBL5887052 0.91 PARP10 (0.39) PARP10PARP15RXRAMAPK1ALDH1A1
SCHEMBL5887098 0.88 PARP10 (0.37) PARP10PARP15RXRAMAPK1ALDH1A1
SCHEMBL5886936 0.88 MAOB (0.39) ALDH1A1CYP1A2CYP3A4USP2CLK4
SCHEMBL5887312 0.88 POLB (0.48) MAPK1ALDH1A1KMT2AMEN1TSHR
SCHEMBL5887577 0.87 ALDH1A1 (0.47) MAPK1ALDH1A1CYP1A2CYP3A4USP2
SCHEMBL5887103 0.82 MAPK14 (0.35) RXRAALDH1A1CYP3A4KMT2ACYP2C9
SCHEMBL5887357 0.77 MAPK14 (0.47) ALDH1A1CYP3A4KMT2AMEN1POLB
SCHEMBL5887013 0.76 TTK (0.40) TSHRMAPT
SCHEMBL5886768 0.76 HPGD (0.47) ALDH1A1CYP3A4KMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US disclosed