SCHEMBL5887103

SCHEMBL5887103

Cc1cc(C(N)=O)ccc1Oc1nc(C)c2ccc(=O)n(-c3ccc(C(N)=O)cc3)c2n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.35
BMX P51813 1/20 0.35
BTK Q06187 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
RXRA P19793 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
KCNH2 Q12809 2/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
GLA P06280 1/20 0.33
NPC1 O15118 1/20 0.32
PIK3R2 O00459 1/20 0.32
KMT2A Q03164 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
OPRM1 P35372 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887454 0.89 PDE4B (0.38) MAPK14SMN1; SMN2LMNAMAPK8
SCHEMBL5887358 0.86 MAPT (0.42) MAPK14LMNAPOLBALDH1A1HSP90AA1
SCHEMBL5886862 0.85 MAPK8 (0.40) SMN1; SMN2LMNAALDH1A1NPC1KMT2A
SCHEMBL5886854 0.85 SMN1; SMN2 (0.43) SMN1; SMN2POLBALDH1A1KMT2A
SCHEMBL5886787 0.83 RORC (0.41) LMNAALDH1A1MAPK8
SCHEMBL5887323 0.83 MAPK14 (0.40) MAPK14MAPK8
SCHEMBL5887252 0.82 PARP10 (0.45) RXRAPOLBKDM4EALDH1A1KMT2A
SCHEMBL5886767 0.82 ALDH1A1 (0.38) SMN1; SMN2RXRAALDH1A1KMT2ACYP3A4
SCHEMBL5887052 0.82 PARP10 (0.39) MAPK14SMN1; SMN2RXRAKDM4EALDH1A1
SCHEMBL5886936 0.79 MAOB (0.39) SMN1; SMN2KDM4EALDH1A1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US claimed
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors PHARMACIA ITALIA S.P.A. 2004-01-15 US claimed
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors TERT, TERF2, TERF2IP MAPK14 1051/4885BMX 1135/4885BTK 3209/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.