SCHEMBL5887406

SCHEMBL5887406

COc1ccc(C2=C(Cl)[CH]CC(c3ccc(Cl)cc3)=C2F)cc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.42
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
ESR1 P03372 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HPGD P15428 1/20 0.37
ALOX5 P09917 1/20 0.35
GLA P06280 1/20 0.35
GCGR P47871 1/20 0.35
MAPK14 Q16539 1/20 0.35
GSK3B P49841 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887461 0.71 NPC1 (0.39) HSP90AA1HSP90AB1NPC1RAB9ASMN1; SMN2
SCHEMBL3947663 0.70 HPGD (0.59) NPC1RAB9ASMN1; SMN2HPGDALOX5
SCHEMBL5887265 0.69 LTA4H (0.49) PTGS1HSP90AA1HSP90AB1ESR1NPC1
SCHEMBL5887165 0.69 NPC1 (0.38) PTGS1HSP90AA1HSP90AB1NPC1RAB9A
SCHEMBL5887087 0.69 RAD51 (0.41) PTGS1ESR1
SCHEMBL5887214 0.68 RAD51 (0.46) ESR1
SCHEMBL2226770 0.68
SCHEMBL154527 0.68
SCHEMBL5886915 0.67 LTA4H (0.49) PTGS1ESR1NPC1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL11293911 0.66 CA1 (0.65) NPC1RAB9ASMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037931-B2 Corticotropin releasing factor moderator; analgesics; drug abruse, drug dependency; schizophrenia JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-02 US disclosed
US-20050026903-A1 CCK-1 receptor modulators JANSSEN PHARMACEUTICA N.V. (BE) 2005-02-03 US disclosed
US-20050020565-A1 Pyrazole compound; gastrointestinal disorders; central nervous system disorders JONES TODD K (US) 2005-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050020565-A1 Pyrazole compound; gastrointestinal disorders; central nervous system disorders CCKAR, CCKBR, NPY1R PTGS1 1104/4885HSP90AA1 2801/4885HSP90AB1 2751/4885
US-20050026903-A1 CCK-1 receptor modulators CCKAR, CCKBR, GLP1R PTGS1 710/4885HSP90AA1 3070/4885HSP90AB1 2876/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.