SCHEMBL5889528

SCHEMBL5889528

O=C(Nc1ccc2[nH]c(C(=O)NCCNCCO)cc2c1)c1ccc2[nH]c(C(=O)Nc3ccc4[nH]c(C(=O)NCCNCCO)cc4c3)cc2c1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PYGL P06737 4/20 0.48
NHERF1 O14745 3/20 0.48
HDAC2 Q92769 2/20 0.48
PLD2 O14939 1/20 0.47
PLD1 Q13393 1/20 0.47
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
ITGB3 P05106 5/20 0.46
ITGA2B P08514 5/20 0.46
MAOA P21397 2/20 0.46
MAOB P27338 2/20 0.46
EGFR P00533 2/20 0.45
PIK3CA P42336 2/20 0.45
AKR1C3 P42330 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5889645 0.95 KDM4E (0.46) PYGLNHERF1HDAC2PLD2PLD1
SCHEMBL5889574 0.90 KDM4E (0.50) NHERF1HDAC2PLD2PLD1KDM4E
SCHEMBL5889512 0.89 HDAC2 (0.50) NHERF1HDAC2PLD2PLD1KDM4E
SCHEMBL5889839 0.86 HDAC2 (0.56) NHERF1HDAC2PLD2PLD1KDM4E
SCHEMBL5896620 0.85 KDM4E (0.50) PYGLNHERF1PLD2PLD1KDM4E
SCHEMBL5889622 0.84 ITGB3 (0.53) PYGLNHERF1HDAC2PLD2PLD1
Hydrochloric Acid SCHEMBL6809892 0.84 HDAC2 (0.44) PYGLNHERF1HDAC2PLD2PLD1
SCHEMBL5889830 0.84 KDM4E (0.57) NHERF1HDAC2PLD2PLD1KDM4E
SCHEMBL5889837 0.83 HDAC2 (0.48) PYGLNHERF1HDAC2PLD2PLD1
SCHEMBL5677265 0.83 ITGB3 (0.54) PYGLNHERF1HDAC2PLD2PLD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7064218-B2 Aromatic compounds and poly(oxyalkylene) containing aromatic compounds possessing antibacterial, antifungal or antitumor activity GENELABS TECHNOLOGIES, INC. (US) 2006-06-20 US disclosed
US-6906103-B2 Compounds possessing antibacterial, antifungal or antitumor activity GENELABS TECHNOLOGIES, INC. (US) 2005-06-14 US disclosed
US-6849713-B2 Compounds possessing antibacterial, antifungal or antitumor activity GENELABS TECHNOLOGIES, INC. (US) 2005-02-01 US disclosed
US-20030212113-A1 Novel aromatic compounds and poly(oxyalkylene) containing aromatic compounds possessing antibacterial, antifungal or antitumor activity GLAXOSMITHKLINE LLC 2003-11-13 US disclosed
WO-2003057212-A1 POLYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL, ANTIFUNGAL OR ANTITUMOR ACTIVITY GENELABS TECHNOLOGIES, INC. (US) 2003-07-17 WO disclosed
US-20030119749-A1 Novel compounds possessing antibacterial, antifungal or antitumor activity SMITHKLINE BEECHAM CORPORATION 2003-06-26 US disclosed
EP-1294713-A2 COMPOUNDS POSSESSING ANTIBACTERIAL, ANTIFUNGAL OR ANTITUMOR ACTIVITY GENELABS TECHNOLOGIES, INC. (US) 2003-03-26 EP disclosed
WO-2002000650-A9 NOVEL COMPOUNDS POSSESSING ANTIBACTERIAL, ANTIFUNGAL OR ANTITUMOR ACTIVITY GENELABS TECH INC (US) 2003-03-06 WO disclosed
US-20020037856-A1 Novel compounds possessing antibacterial, antifungal or antitumor activity GENELABS TECHNOLOGIES, INC. 2002-03-28 US disclosed
WO-2002000650-A2 NOVEL COMPOUNDS POSSESSING ANTIBACTERIAL, ANTIFUNGAL OR ANTITUMOR ACTIVITY GENELABS TECHNOLOGIES, INC. (US) 2002-01-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030119749-A1 Novel compounds possessing antibacterial, antifungal or antitumor activity CYP51A1, MCL1, ERG28 PYGL 2695/4885NHERF1 1638/4885HDAC2 1132/4885
US-20020037856-A1 Novel compounds possessing antibacterial, antifungal or antitumor activity CYP51A1, MCL1, ERG28 PYGL 2695/4885NHERF1 1638/4885HDAC2 1132/4885
US-20030212113-A1 Novel aromatic compounds and poly(oxyalkylene) containing aromatic compounds possessing antibacterial, antifungal or antitumor activity TYR, CYP51A1, ODC1 PYGL 3731/4885NHERF1 2040/4885HDAC2 2108/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.