SCHEMBL5951968

SCHEMBL5951968

CC1Cc2cccc(-c3cccc(-c4ccccc4)c3)c2C1=O

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 0.54
BRD4 O60885 2/20 0.46
CREBBP Q92793 2/20 0.46
HTR1A P08908 1/20 0.42
DRD2 P14416 1/20 0.42
HTR7 P34969 1/20 0.42
EDNRB P24530 1/20 0.39
EDNRA P25101 1/20 0.39
TDP2 O95551 1/20 0.38
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
MAOA P21397 2/20 0.37
MAOB P27338 2/20 0.37
HDAC4 P56524 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC8 Q9BY41 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5951620 0.94 ACHE (0.54) ACHEBRD4CREBBPHTR1ADRD2
SCHEMBL5952527 0.91 ACHE (0.57) ACHEBRD4CREBBPHTR1ADRD2
SCHEMBL5509273 0.91 ACHE (0.61) ACHEBRD4CREBBPHTR1ADRD2
Dimethylamine SCHEMBL7161154 0.87 ACHE (0.56) ACHEBRD4CREBBPHTR1ADRD2
SCHEMBL5952266 0.85 ACHE (0.50) ACHEMAOAMAOB
SCHEMBL5951689 0.85 ACHE (0.57) ACHEBRD4CREBBPHTR1ADRD2
SCHEMBL5951226 0.84 TDP2 (0.52) ACHETDP2MAOAMAOB
SCHEMBL5952829 0.84 ACHE (0.49) ACHEBRD4HTR1ADRD2HTR7
SCHEMBL5951118 0.83 ACHE (0.51) ACHEMAOAMAOBHDAC4HDAC2
SCHEMBL5952210 0.82 ACHE (0.46) ACHEHTR1ADRD2HTR7MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7038070-B2 Preparation of preparing substituted indanones BASELL POLYOLEFINE GMBH (DE) 2006-05-02 US disclosed
US-6963017-B2 Preparation of preparing substituted indanones BASELL POLYOLEFINE GMBH (DE) 2005-11-08 US disclosed
EP-0968158-B1 METHOD OF PREPARING SUBSTITUTED INDANONES, THE SUBSTITUTED INDANONES AND METALLOCENES PREPARED THEREFROM BASELL POLYOLEFINE GMBH (DE) 2005-08-10 EP disclosed
US-20050033076-A1 Preparation of preparing substituted indanones EQUISTAR CHEMICALS, LP 2005-02-10 US disclosed
US-20030009046-A1 Preparation of preparing substituted indanones EQUISTAR CHEMICALS, LP 2003-01-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050033076-A1 Preparation of preparing substituted indanones CYP1A2, CYP2J2, IDH3A ACHE 839/4885BRD4 3097/4885CREBBP 2331/4885
US-20030009046-A1 Preparation of preparing substituted indanones CYP1A2, CYP1B1, CYP1A1 ACHE 820/4885BRD4 3045/4885CREBBP 2466/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.