SCHEMBL5960985

SCHEMBL5960985

Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc(N)c(C(O)c2cccc(Cl)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
RORC P51449 10/20 0.52
FNTA P49354 5/20 0.51
FNTB P49356 5/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4373341 0.82 FNTA (0.46) RORCFNTAFNTB
SCHEMBL4370247 0.82 FNTA (0.47) RORCFNTAFNTB
SCHEMBL4381109 0.78 FNTA (0.54) RORCFNTAFNTB
SCHEMBL4381517 0.77 FNTA (0.50) FNTAFNTB
SCHEMBL4052433 0.75 RORC (0.55) RORCFNTAFNTB
SCHEMBL5776979 0.71 RORC (0.63) RORCFNTAFNTB
SCHEMBL5781212 0.71 FNTA (0.67) RORCFNTAFNTB
SCHEMBL5549507 0.69 RORC (0.47) RORCFNTAFNTB
SCHEMBL6586870 0.69 FNTA (0.77) RORCFNTAFNTB
SCHEMBL5783176 0.69 FNTA (0.69) RORCFNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7153958-B2 Farnesyl transferase inhibiting benzoheterocyclic derivatives JANSSEN PHARMACEUTICA N.V. (BE) 2006-12-26 US disclosed
US-20040034218-A1 Farnesyl transferase inhibiting benzoheterocyclic derivatives JANSSEN PHARMACEUTICA N.V. (BE) 2004-02-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040034218-A1 Farnesyl transferase inhibiting benzoheterocyclic derivatives FNTA, FNTB, RCE1 RORC 209/4885FNTA 1/4885FNTB 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.