SCHEMBL5963640

SCHEMBL5963640

CCOC(=O)C(Br)(Br)CC(=O)c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.64
NPSR1 Q6W5P4 1/20 0.64
KMT2A Q03164 4/20 0.53
NPC1 O15118 4/20 0.53
MEN1 O00255 3/20 0.53
PIN1 Q13526 1/20 0.49
ALDH1A1 P00352 4/20 0.46
MAPT P10636 3/20 0.45
PTPN1 P18031 1/20 0.44
GSK3B P49841 1/20 0.44
RAB9A P51151 3/20 0.44
GAA P10253 2/20 0.44
GLA P06280 1/20 0.43
RECQL P46063 1/20 0.43
MMP8 P22894 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
KDM4E B2RXH2 1/20 0.42
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12121920 0.85 POLB (0.66) POLBNPSR1KMT2ANPC1MEN1
SCHEMBL29492080 0.81 POLB (0.69) POLBNPSR1KMT2ANPC1MEN1
SCHEMBL29110257 0.80 POLB (0.59) POLBNPSR1KMT2ANPC1MEN1
SCHEMBL5036126 0.77 ALDH1A1 (0.66) POLBNPSR1KMT2ANPC1MEN1
SCHEMBL5743401 0.76 PIN1 (0.42) POLBNPSR1KMT2AMEN1PIN1
SCHEMBL5964067 0.76 GSK3B (0.56) POLBNPSR1KMT2ANPC1MEN1
SCHEMBL7791515 0.76 POLB (0.56) POLBNPSR1KMT2ANPC1MEN1
SCHEMBL8679766 0.76 PIN1 (0.51) POLBNPSR1KMT2ANPC1MEN1
SCHEMBL1925793 0.75 POLB (0.58) POLBNPSR1KMT2ANPC1MEN1
SCHEMBL11117141 0.75 POLB (0.54) POLBNPSR1KMT2ANPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1143959-B1 ANTIFUNGAL ACTIVITY OF DICATIONIC MOLECULES UNIV NORTH CAROLINA (US) 2006-11-02 EP disclosed
EP-1685836-A2 Antifungal activity of dicationic molecules UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2006-08-02 EP disclosed
EP-0792271-B1 FURAN DERIVATIVES FOR INHIBITING PNEUMOCYSTIS CARINII PNEUMONIA, GIARDIA LAMBLIA AND CRYPTOSPORIDIUM PARVUM UNIV GEORGIA STATE RES FOUND (US) 2002-02-27 EP disclosed
US-6326395-B1 AMIDINE OR AMIDE SUBSTITUTED FURAN DERIVATIVES DUKE UNIVERSITY 2001-12-04 US disclosed
EP-1143959-A2 ANTIFUNGAL ACTIVITY OF DICATIONIC MOLECULES UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2001-10-17 EP disclosed
WO-2000015212-A2 ANTIFUNGAL ACTIVITY OF DICATIONIC MOLECULES THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2000-03-23 WO disclosed
EP-0792271-A1 FURAN DERIVATIVES FOR INHIBITING PNEUMOCYSTIS CARINII PNEUMONIA, GIARDIA LAMBLIA AND CRYPTOSPORIDIUM PARVUM GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 1997-09-03 EP disclosed
US-5602172-A USING A 2,5-DIPHENYLFURAN COMPOUND THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1997-02-11 US disclosed
WO-1996015126-A1 FURAN DERIVATIVES FOR INHIBITING PNEUMOCYSTIS CARINII PNEUMONIA, GIARDIA LAMBLIA AND CRYPTOSPORIDIUM PARVUM GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 1996-05-23 WO disclosed