SCHEMBL5981399

SCHEMBL5981399

Cc1ccccc1-c1ccc2c(c1C(=O)O)OC(c1ccccc1)(c1ccccc1)O2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 8/20 0.39
LDHA P00338 1/20 0.39
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
HTT P42858 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
HPGD P15428 1/20 0.35
MYC P01106 1/20 0.35
MCL1 Q07820 2/20 0.34
NR1H4 Q96RI1 1/20 0.33
APAF1 O14727 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
TACR1 P25103 1/20 0.33
RPA1 P27694 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9040225 0.74 CNR1 (0.42) CNR1CYP1A2MYCALDH1A1
SCHEMBL25137230 0.73 CNR1 (0.39) CNR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9074662 0.70 CNR1 (0.44) CNR1CYP1A2NPSR1HPGDALDH1A1
SCHEMBL4860502 0.69 ALOX5 (0.43) CNR1CYP2C9HPGDMYCALDH1A1
SCHEMBL4466643 0.69 CNR1 (0.44) CNR1LDHAALDH1A1
SCHEMBL6679648 0.69 MYC (0.55) LDHACYP3A4CYP2C9HTTL3MBTL1
SCHEMBL4862066 0.69 CNR1 (0.40) CNR1CYP3A4CYP2C9CYP2C19NPSR1
SCHEMBL6226020 0.68 CNR1 (0.64) CNR1LDHAMYCALDH1A1
SCHEMBL5982862 0.68 CNR1 (0.33) CNR1NPSR1
SCHEMBL8285530 0.68 CNR1 (0.44) CNR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697394-A2 COMT INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2006-09-06 EP disclosed
WO-2005058228-A2 COMT INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-30 WO disclosed