SCHEMBL5983310

SCHEMBL5983310

CN(c1cccc(NC(=O)c2ccncc2)c1)C1CCNCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 3/20 0.51
LMNA P02545 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
KCNK9 Q9NPC2 1/20 0.49
P2RY14 Q15391 1/20 0.46
HTT P42858 2/20 0.46
RXFP1 Q9HBX9 1/20 0.44
TRPV1 Q8NER1 1/20 0.44
GAA P10253 1/20 0.43
FDPS P14324 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KDM4E B2RXH2 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
MAPK1 P28482 2/20 0.42
ALDH1A1 P00352 1/20 0.42
RAB9A P51151 1/20 0.42
POLB P06746 1/20 0.41
ITGA2B P08514 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5982835 0.86 MEN1 (0.53) KCNK3MEN1KMT2AKCNK9HTT
Hydrochloric Acid SCHEMBL5983863 0.80 RAB9A (0.47) LMNASMN1; SMN2HTTMAPK1ALDH1A1
Hydrochloric Acid SCHEMBL5983348 0.79 SMN1; SMN2 (0.53) KCNK3SMN1; SMN2MEN1KMT2AKCNK9
Hydrochloric Acid SCHEMBL5983919 0.78 F2R (0.52) LMNAMEN1KMT2ARXFP1L3MBTL1
Hydrochloric Acid SCHEMBL5983763 0.78 KCNK3 (0.49) KCNK3MEN1KMT2AKCNK9RXFP1
Hydrochloric Acid SCHEMBL5983539 0.77 PTGS1 (0.56) KCNK3MEN1KMT2AKCNK9RXFP1
Hydrochloric Acid SCHEMBL5983492 0.77 ALDH1A1 (0.43) MEN1KMT2AL3MBTL1ALDH1A1RAB9A
SCHEMBL2550898 0.76 DDB1 (0.36)
SCHEMBL5983644 0.76 RXFP1 (0.43) RXFP1
Hydrochloric Acid SCHEMBL5983356 0.76 TLR7 (0.48) SMN1; SMN2GAAL3MBTL1KDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663971-A1 SUBSTITUTED 2-CARBONYLAMINO-6-PIPERIDINAMINOPYRIDINES AND SUBSTITUTED 1-CARBONYLAMINO-3-PIPERIDINAMINOBENZENES AS 5-HT1F AGONISTS Eli Lilly and Company (US) 2006-06-07 EP disclosed
WO-2005035499-A1 SUBSTITUTED 2-CARBONYLAMINO-6-PIPERIDINAMINOPYRIDINES AND SUBSTITUTED 1-CARBONYLAMINO-3-PIPERIDINAMINOBENZENES AS 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2005-04-21 WO disclosed