SCHEMBL5987962

SCHEMBL5987962

CC(C)(C)OC(=O)NCc1nc(C#N)no1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.39
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.37
KDM4A O75164 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.35
CTSS P25774 3/20 0.35
CTSK P43235 3/20 0.35
BCHE P06276 1/20 0.34
GFER P55789 1/20 0.34
CACNA1H O95180 1/20 0.34
CACNA1B Q00975 1/20 0.34
CACNA1C Q13936 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6467979 0.80 KCNJ1 (0.43) CYP1A2KDM4ELMNAHTTKDM4A
SCHEMBL8279808 0.78 MAPT (0.50) LMNAMAPT
SCHEMBL6652772 0.78 MAPT (0.30) TDP1MAPT
SCHEMBL411489 0.77 CACNA1H (0.42) CYP1A2KDM4ELMNAHTTKDM4A
SCHEMBL7984088 0.75 HTT (0.39) CYP1A2KDM4ELMNAHTTKDM4A
SCHEMBL29523683 0.74 HTT (0.46) KDM4ELMNAHTTNPSR1TDP1
SCHEMBL5987499 0.74 HTT (0.38) CYP1A2KDM4ELMNAHTTKDM4A
SCHEMBL6476856 0.72 L3MBTL1 (0.46) KDM4ELMNAKDM4ANPSR1L3MBTL1
SCHEMBL14679174 0.72 MAPT (0.66) MAPT
SCHEMBL4516428 0.72 GPR119 (0.53) KDM4ELMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7144902-B1 Prodrugs of thrombin inhibitors ABBOTT GMBH & CO. KG (DE) 2006-12-05 US disclosed
US-6740647-B1 AMIDINES AND HYDROXYAMIDINE DERIVATIVES ABBOTT GMBH & CO., KG (DE) 2004-05-25 US disclosed
EP-1051431-A1 THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-11-15 EP disclosed
US-6114358-A Thrombin inhibitors BASF AKTIENGESELLSCHAFT (DE) 2000-09-05 US disclosed
WO-1999037668-A1 THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-07-29 WO disclosed