SCHEMBL5988264

SCHEMBL5988264

Cc1ccc2c(Sc3ccccc3C(=O)N(C)C)c[nH]c2c1.Cc1cccc(C(N)=O)c1C

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
HPGD P15428 1/20 0.40
SLC6A4 P31645 2/20 0.37
IDO1 P14902 2/20 0.36
NR4A2 P43354 1/20 0.36
GFER P55789 1/20 0.33
NPC1 O15118 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
ATM Q13315 1/20 0.33
KDR P35968 2/20 0.32
CDK4 P11802 1/20 0.32
CCND1 P24385 1/20 0.32
STAT3 P40763 1/20 0.32
SLC6A2 P23975 1/20 0.31
SLC6A3 Q01959 1/20 0.31
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1399258 0.89 ALDH1A1 (0.49) ALDH1A1MEN1MAPTKMT2AHPGD
SCHEMBL1399397 0.78 ALDH1A1 (0.49) ALDH1A1MEN1MAPTKMT2AHPGD
SCHEMBL1399233 0.77 ALDH1A1 (0.48) ALDH1A1MEN1MAPTKMT2AHPGD
SCHEMBL1399426 0.77 ALDH1A1 (0.64) ALDH1A1MEN1MAPTKMT2AHPGD
SCHEMBL1399377 0.77 ALDH1A1 (0.46) ALDH1A1MEN1MAPTKMT2AHPGD
SCHEMBL1399458 0.76 GFER (0.52) ALDH1A1MEN1MAPTKMT2AHPGD
SCHEMBL1399287 0.76 HPGD (0.48) ALDH1A1MEN1MAPTKMT2AHPGD
SCHEMBL1399417 0.75 MAPT (0.47) ALDH1A1MEN1MAPTKMT2AHPGD
SCHEMBL1399418 0.74 BRPF1 (0.48) ALDH1A1MEN1MAPTKMT2AHPGD
SCHEMBL1399354 0.71 ALDH1A1 (0.64) ALDH1A1MEN1MAPTKMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1701940-A1 2-(1H-INDOLYLSULFANYL)-BENZYL AMINE DERIVATIVES AS SSRI H.Lundbeck A/S (DK) 2006-09-20 EP disclosed
WO-2005061455-A1 2-(1H-INDOLYLSULFANYL)-BENZYL AMINE DERIVATIVES AS SSRI H. LUNDBECK A/S (DK) 2005-07-07 WO disclosed